| Cat. No. |
Product Name |
Information |
| PC-20399 |
SAN4825
ADPR-cyclase inhibitor
|
SAN4825 is a selective small-molecule inhibitor of cardiac ADP-ribosyl cyclase (ADPR cyclase) with IC50 of 0.13 uM. |
| PC-20389 |
Dantrolene
Glutathione reductase inhibitor, RyR antagonist
|
Dantrolene (F368) is a muscle relaxant, non-competitively inhibitor of human erythrocyte glutathione reductase with Ki and IC50 values are 111.6 μM and 52.3 μM, respectively. |
| PC-20384 |
Sulfosuccinimidyl oleate sodium
CD36 inhibitor
|
Sulfosuccinimidyl oleate sodium (SSO) is an irreversible inhibitor of the fatty acid translocase CD36, inhibits fatty acid transport (FAT) into cells. |
| PC-20371 |
PIP5K inhibitor 20
PIP5K inhibitor
|
PIP5K inhibitor 20 is a potent, selective pan-PIP5K inhibitor with IC50 values of 58, 46 and 39 nM for PIP5Kα, PIP5Kβ and PIP5Kγ, respectively. |
| PC-20346 |
SYNTi
Syndecan/syntenin inhibitor
|
SYNTi is a small molecule PDZ domain inhibitor targeting the syndecan/syntenin protein-protein interaction with IC50 of 400 nM. |
| PC-20337 |
TDRL-551
RPA inhibitor
|
TDRL-551 (TDRL551) is a small molecule Replication Protein A (RPA) inhibitor targeting the Replication Protein A-DNA interaction with IC50 of 18 uM. |
| PC-20325 |
HTL0041178
GPR52 agonist
|
HTL0041178 is a potent GPR52 agonist with EC50 of 27.5 nM (human or rat GPR52). |
| PC-20321 |
BC-K-YH16899
KRS-67LR inhibitor
|
BC-K-YH16899 (YH16899) is a specific small molecule inhibitor of prometastatic lysyl-tRNA synthetase-laminin receptor interaction (KRS-67LR PPI), suppresses cancer metastasis. |
| PC-20318 |
Secdin
ARF-GEF inhibitor
|
Secdin is a small-molecule inhibitor of Arabidopsis thaliana ADP-ribosylation factor (ARF)-guanine nucleotide exchange factors (GEFs), impaires both hypocotyl and root growth in young Arabidopsis seedlings with IC50 of 4 uM. |
| PC-20313 |
SJ572946
BAK activator
|
SJ572946 is a small molecule BAK activator, binds to the activation groove of BAK and selectively triggers BAK activation over that of BAX in liposome and mitochondrial permeabilization assays. |
| PC-20306 |
ELOVL6 inhibitor Compound B
ELOVL6 inhibitor
|
ELOVL6 inhibitor Compound B is a potent and selective ELOVL6 inhibitor with IC50 of 85 and 38 nM for human and mouse ELOVL6, respectively. |
| PC-20305 |
ELOVL6 inhibitor 37
ELOVL6 inhibitor
|
ELOVL6 inhibitor 37 (ELOVL6-IN-2) is a potent, selective inhibitor of elongase of long-chain fatty acids family 6 (ELOVL6) with IC50 of 8.9 and 31 nM for human and mouse ELOVL6, respectively. |
