CRAC Channel (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-22078	MRS1845 SOCE channel inhibitor, Orai1 inhibitor	MRS1845 is a selective store-operated Ca2+ channel (SOC) Orai1 inhibitor, inhibits SOC channel-dependent elevations of calcium with IC50 of 1.7 uM in HL-60 cells.
PC-38432	Zegocractin Orai1 channel inhibitor	Zegocractin (CM-4620, CM-128) is a selective small molecule CRAC (Orai1) channel inhibitor, inhibits Orai1/STIM1-mediated Ca2+ currents and Orai2/STIM1-mediated currents with IC50 of 120 nM and 900 nM, respectively.
PC-43089	GSK-5498A CRAC channel inhibitor	GSK-5498A is a potent, selective small molecule blocker of Calcium-Release Activated Calcium (CRAC) channel with IC50 of 1 uM.
PC-60224	Synta66 CRAC channel inhibitor	Synta66 (Synta-66, GSK1349571A) is a potent, selective CRAC channel Orai1 blocker with IC50 of 3 uM.
PC-70096	GSK-7975A Orai1 inhibitor	GSK-7975A (GSK7975A) is a selective CRAC channel essential pore subunit Orai1 blocker that inhibits store-operated Ca(2+) entry (SOCE) with IC50 of 3.4 uM.
PC-42271	YM-58483 CRAC channel inhibitor	YM-58483 is a potent store-operated Ca2+ entry blocker and CRAC channel inhibitor with IC50 of 100 nM.

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