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Cat. No. Product Name Information
PC-38552

EC23

EC23 (AGN190205) is a photostable synthetic retinoid and analog of ATRA, potently induces neural differentiation in human pluripotent embryonic stem cells.
PC-38546

DL5H3

DL5H3 is a bioactive compound with antiasthmatic activity.
PC-38539

KLH45

DDHD2 inhibitor

KLH45 is a potent, selective and in vivo-active serine hydrolase DDHD2 inhibitor with IC50 of 1.3 nM, shows excellent selectivity against other serine hydrolases with exception of ABHD6.
PC-38530

NCGC607

GCase activator

NCGC00241607 (NCGC607) is a small-molecule noninhibitory chaperone of glucocerebrosidase (GCase), successfully chaperoned the mutant enzyme, restored GCase activity and protein levels, and reduced glycolipid storage in neurons.
PC-38529

pythiDC

CP4H1 inhibitor

pythiDC is a small molecule inhibitor of human CP4H1 with IC50 of 4.0 uM, inhibits CP4H activity in cultured cells at concentrations that do not cause iron deficiency.
PC-38525

ML198

GCase chaperone

ML198 is a non-inhibitory chaperone of glucocerebrosidase (GCase) enzyme, does not inhibit the enzyme’s action, but can facilitate its translocation to the lysosome.
PC-38518

MSBN

MSBN is a highly selective fluorogenic probe for thiols, selectively imaging thiols in live cells and specifically label protein thiols with a turn-on signal to determine diverse reversible protein thiol modifications.
PC-38516

GSK106

PAD4 inhibitor

GSK106 is an inactive control for the selective PAD4 inhibitors, GSK484 and GSK199.
PC-38515

Creatine riboside

Creatine riboside is a metabolite standard and classifier of lung cancer status in all and stage I–II cases, important for early detection, and also associated with worse prognosis in stage I–II lung cancer.
PC-38501

MrgX1 modulator 8e

MrgX1 modulator

MrgX1 inhibitor 8e is a potent, allosteric modulator of MrgX1 with EC50 of 13 nM, shows improved potency and microsomal stability than ML382.
PC-38497

UNC7467

IP6K inhibitor

UNC7467 is a potent, selective inositol hexakisphosphate kinase (IP6K) inhibitor with IC50 values of 8.9 nM (IP6K1), 4.9 nM (IP6K2) and 1320 nM (IP6K3).
PC-38482

CYM2503

GalR2 PAM

CYM2503 is a putative galanin receptors type 2 (GalR2) positive allosteric modulator, concentration-dependently potentiates galanin (100 nM) stimulated IP1 accumulation in HEK293-GalR2 cells with EC50 of 0.69 uM, efficacy of 9.7-fold potentiation.

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