| Cat. No. |
Product Name |
Information |
| PC-22666 |
Myeloperoxidase inhibitor RL6
Myeloperoxidase inhibitor
|
Myeloperoxidase inhibitor RL6 is a potent, reversible inhibitor of myeloperoxidase (MPO) and hypochlorous acid (HOCl) scavenger, inhibits neutrophil extracellular trap release (NETosis). |
| PC-22644 |
TAK-683
KISS1R agonist
|
TAK-683 is a potent and full KISS1R (metastin receptor) agonist and kisspeptin analogue with IC50 of 3 pM in radioimmunoassay. |
| PC-22643 |
TAK-683 acetate
KISS1R agonist
|
TAK-683 acetate is a potent and full KISS1R (metastin receptor) agonist and kisspeptin analogue with IC50 of 3 pM in radioimmunoassay. |
| PC-22642 |
TAK-448 acetate
KISS1R agonist
|
TAK-448 (MVT-602) acetate is a potent and full KISS1R (metastin receptor) agonist and kisspeptin analogue with IC50 of 3 pM in radioimmunoassay. |
| PC-22636 |
Delphinidin chloride
Hyaluronidase inhibitor
|
Delphinidin chloride is a natural plant compound found in fruits and vegetables, a potent hyaluronidase inhibitor, increases high molecular weight hyaluronic acid (HMW-HA) and inhibits cancer metastasis. |
| PC-22628 |
GGTI-2154 hydrochloride
GGTase I inhibitor
|
GGTI-2154 hydrochloride is a potent, selective inhibitor geranylgeranyltransferase I (GGTase I) with IC50 f 21 nM, >250-fold selective over FTase. |
| PC-22627 |
GGTI-2154
GGTase I inhibitor
|
GGTI-2154 is a potent, selective inhibitor geranylgeranyltransferase I (GGTase I) with IC50 f 21 nM, >250-fold selective over FTase. |
| PC-22593 |
UNC10245380
CIB1 inhibitor
|
UNC10245380 (UNC5380) is a small molecule ligand/inhibitor of Calcium and Integrin Binding protein 1 (CIB1) with IC50 of 8.0 uM in TR-FRET displacement assay, selectively kills CIB1 depletion-sensitive TNBC cells. |
| PC-22571 |
TMLB-C16
B3GAT3 inhibitor
|
TMLB-C16 is a potent beta-1,3-glucuronosyltransferase (B3GAT3) inhibitor with KD of 3.96 uM, suppresses proliferation and migration in HCC cells. |
| PC-22540 |
YK-4-279
EWS-FLI1 inhibitor
|
YK-4-279 is a specific small molecule inhibitor of EWS-FLI1 interaction with RNA helicase A with SPR KD of 9.48 uM for EWS-FLI1, reduces EWS-FLI1 functional activity, also reduces EWS-FLI1 modulated transcription. |
| PC-22489 |
UR778Br
IQGAP1 inhibitor
|
UR778Br is a potent small molecule inhibitor of scaffolding protein IQGAP1, taregting the IQGAP1-GRD domain, selectively inhibits growth of human acute myeloid leukemia. |
| PC-22470 |
PW0729
GPR52 agonist
|
PW0729 is a potent, selective, G protein-biased agonist of orphan GPR52 with EC50 of 47 nM in cAMP assay, Emax=143%. |
