Cat. No. |
Product Name |
Information |
PC-73150 |
Eptifibatide acetate
Glycoprotein IIb/IIIa inhibitor
|
Eptifibatide acetate is a synthetic homodetic cyclic peptide, inhibits platelet aggregation by selectively blocking the platelet glycoprotein IIb/IIIa receptor. |
PC-73149 |
DLin-MC3-DMA
|
DLin-MC3-DMA is an ionizable amino lipid (apparent pKa = 6.44) that has been used in combination with other lipids in the formation of lipid nanoparticles. |
PC-73143 |
MCU-i11
MICU1 inhibitor
|
MCU-i11 is a specific MICU1 targeting compound that negative modulate mitochondrial Ca2+ uptake. |
PC-73142 |
MCU-i4
MICU1 inhibitor
|
MCU-i4 is a specific MICU1 targeting compound that negative modulate mitochondrial Ca2+ uptake. |
PC-73139 |
ASN90
O-GlcNAcase inhibitor
|
ASN90 is a potent, selective, substrate-competitive O-GlcNAcase (OGA) inhibitor with IC50 of 10.2 nM. |
PC-73138 |
KVD900
Plasma kallikrein inhibitor
|
Sebetralstat (KVD900) is a potent, selective, competitive and reversible inhibitor of human plasma kallikrein (PKa) enzyme with Ki of 3.02 nM. |
PC-73136 |
Naphthyridine-azaquinolone
Slipped-CAG DNA binder
|
Naphthyridine-azaquinolone (NA) is a specific small molecule that specifically binds slipped-CAG DNA intermediates of expansion mutations. |
PC-73135 |
PGAM1 inhibitor KH3
PGAM1 inhibitor
|
PGAM1 inhibitor KH3 is a potent, allosteric small molecule inhibitor of phosphoglycerate mutase 1 (PGAM1) with IC50 of 105 nM. |
PC-73129 |
HG106
SLC7A11 inhibitor
|
HG106 (HG 106) is a potent, selective SLC7A11 inhibitor, selectively kills KRAS-mutant lung adenocarcinoma (LUAD) cells. |
PC-73123 |
CU-76
cGAS inhibitor
|
CU-76 (cGAS inhibitor CU-76) is a small-molecule human cGAS (hcGAS) inhibitor with IC50 of 0.24 uM. |
PC-73115 |
AZD9898
LTC4S inhibitor
|
AZD9898 (AZD-9898) is a highly potent, selective and oral inhibitor of leukotriene C4 synthase (LTC4S) with IC50 of 0.28 nM. |
PC-73111 |
S-181
GCase activator
|
S-181 (S 181) is a specific small-molecule activator (modulator) of β-glucocerebrosidase (GCase) with AC50 of 1.49 uM and a maximum activation of 780%. |