| Cat. No. |
Product Name |
Information |
| PC-45056 |
USP7-IN-1
USP7 inhibitor
|
USP7-IN-1 is a novel selective and reversible inhibitor of USP7 with IC50 of 33 uM. |
| PC-46007 |
SJB3-019A
USP1 inhibitor
|
SJB3-019A is a potent ubiquitin-specific protease USP1 inhibitor with IC50 of 78.1 nM, 5 times more potent than SJB2-043 in promoting ID1 degradation and cytoxicity in K562 cells. |
| PC-24052 |
USP1 inhibitor 38-P2
USP1 inhibitor
|
USP1 inhibitor 38-P2 is a potent, selective, reversible, and noncompetitive ubiquitin-specific protease 1 (USP1) inhibitor with IC50 of 3.8 nM (USP1-UAF1). |
| PC-23952 |
U4-I05
USP4 inhibitor
|
U4-I05 is a specific small molecule USP4 inhibitor (KD=239 nM) that inhibits USP4 deubiquitinating enzyme activity, inhibits stemness characteristics in CRC cells. |
| PC-23862 |
USP30i-3
USP30 inhibitor
|
USP30i-3 is a potent, selective small molecule USP30 inhibitor with IC50 of 21 nM, selective over other DUBs (IC50=250->3000 nM) with exception of USP6 (IC50=60 nM). |
| PC-23861 |
USP30i-37
USP30 inhibitor
|
USP30i-37 is a potent, selective small molecule USP30 inhibitor with IC50 of 48 nM, selective over other DUBs (IC50=400->3000 nM) with exception of USP6 (IC50=95 nM). |
| PC-23860 |
ST-539
USP30 inhibitor
|
ST-539 is a potent mitophagy inducer and selective USP30 inhibitor (IC50=0.37 uM), does not inhibit USP1, 8 and 9 at 10 uM. |
| PC-23859 |
MTX652
USP30 inhibitor
|
MTX652 is potent and selective inhibitor of deubiquitinating enzyme USP30. |
| PC-23737 |
USP30 inhibitor 11
USP30 inhibitor
|
USP30 inhibitor 11 is a selective and potent ubiquitin specific peptidase 30 (USP30) inhibitor with IC50 of <10 nM. |
| PC-23736 |
USP30-I-1
USP30 inhibitor
|
USP30-I-1 is a potent, selective and covalent inhibitor of mitochondrial deubiquitinating (DUB) enzyme USP30 with IC50 of 94 nM, shows no significant activity against other 40 endogenous DUBs. |
| PC-23143 |
IsoLiPro
USP11 inhibitor
|
IsoLiPro is a novel small molecule USP11 inhibitor, reduces the USP11 protein level and suppressesthe USP11-mediated substrate deubiquitination. |
| PC-23140 |
LN-439A
BAP1 inhibitor
|
LN-439A is a small molecule BRCA1-associated protein 1 (BAP1) inhibitor by binding to the catalytic pocket of BAP1, leading to the ubiquitination and degradation of Krüppel-like factor 5 (KLF5), inhibits proliferation and migration of BLBC cells. |
