| Cat. No. |
Product Name |
Information |
| PC-61935 |
USP7i-1
USP7 inhibitor
|
USP7i-1 (USP7-IN-1) is a potent, selective USP7 inhibitor with IC50 of 77 uM. |
| PC-61934 |
USP10-IN-3
USP10 inhibitor
|
USP10-IN-3 is a HBX19818 analog, potent and selective USP10 inhibitor, but does not inhibit USP7 (IC50>100 uM). |
| PC-61933 |
USP10-IN-9
USP10 inhibitor
|
USP10-IN-9 is a HBX19818 analog, selective USP10 inhibitor with IC50 similar to HBX19818, but does not inhibit USP7 (IC50>100 uM).. |
| PC-61702 |
TCID
UCHL3 inhibitor
|
TCID is a selective ubiquitin C-terminal hydrolase-L3 (UCH-L3) inhibitor with IC50 of 0.6 uM, displays >100-fold selectivity over UCH-L1. |
| PC-61626 |
BC-1471
STAMBP inhibitor
|
BC-1471 is a selective, small-molecule deubiquitinase STAM-binding protein (STAMBP) inhibitor (IC50=0.33 uM) that interrupts STAMBP-Ub-NALP7 interaction. |
| PC-61303 |
EOAI3402143
Usp9x/Usp24 inhibitor
|
EOAI3402143 (Deubiquitinase inhibitor G9, EOAI 3402143) is a novel covalent deubiquitinase Usp9x/Usp24 inhibitor (IC50=1.6 uM). |
| PC-61234 |
IU-1
USP14 inhibitor
|
IU-1 (USP14 inhibitor IU1) is a specific, small molecule inhibitor of deubiquitinating enzyme USP14 with IC50 of 4-5 uM. |
| PC-60494 |
XL188
USP7 inhibitor
|
XL188 (XL-188) is a potent, selective, non-covalent active-site inhibitor of USP7 with IC50 of 90 nM and 193 nM for USP7 full length enzyme and catalytic domain, respectively. |
| PC-60089 |
GNE-6776
USP7 inhibitor
|
GNE-6776 is a novel potent, specific, non-covalent, orally bioavailable USP7 inhibitor with IC50 of 1.34 uM. |
| PC-60088 |
FT-671
USP7 inhibitor
|
FT-671 is a novel potent, specific, non-covalent USP7 inhibitor with Kd of 65 nM (USP7 catalytic domain). |
| PC-60087 |
FT827
USP7 inhibitor
|
FT827 is a novel potent, specific, covalent USP7 inhibitor with Kd of 7.8 uM (USP7 catalytic domain). |
| PC-60026 |
USP25 and 28 inhibitor AZ2
USP25/USP28 inhibitor
|
USP25 and 28 inhibitor AZ2 is a potent, selective, dual USP25/28 inhibitor with IC50 of 0.9/0.9 uM, respectively. |
