| Cat. No. |
Product Name |
Information |
| PC-20796 |
BK50118-C
USP13 inhibitor
|
BK50118-C is a potent small molecule inhibitor of ubiquitin-specific protease-13 (USP13) with IC50 of 0.42 nM. |
| PC-20656 |
b-AP15
USP14 inhibitor
|
b-AP15 (bAP15, NSC 687852) is a specific inhibitor of ubiquitin-specific-processing protease 14 (USP14) and ubiquitin carboxyl-terminal hydrolase isozyme L5 (UCHL5), inhibits DUB activity in purified 19S proteasomes with IC50 of 2.1 uM. |
| PC-20480 |
Neutral Red
USP4 inhibitor
|
Neutral Red is a nitrogenous pH-indicator that can stains lysosomes red, also is a selective, uncompetitive USP4 inhibitor with IC50 of 50 uM. |
| PC-20472 |
IU1-206
USP14 inhibitor
|
IU1-206 is a IU1 derivative with more potent activity against USP14, 10-fold more potent than IU1 and is comparable to the IU1-47. |
| PC-20403 |
PR-619
DUBs inhibitor
|
PR-619 (PR619) is a broad-spectrum, reversible deubiquitinating enzymes (DUBs), inhibits USP4, USP8, USP7, USP2, and USP5 with IC50 of 3.93, 4.9, 6.86, 7.2, and 8.61 uM, respectively. |
| PC-20202 |
HBX41108
USP7 inhibitor
|
HBX41108 is a specific small-molecule inhibitor of USP7/HAUSP ubiquitin protease with IC50 of 424 nM for inhibition of Ub-AMC hydrolysis by USP7. |
| PC-20190 |
USP14 inhibitor 3
USP14 inhibitor
|
USP14-IN-3 is a specific small molecule USP14 inhibitor with IC50 of <0.5 uM. |
| PC-20189 |
USP14 inhibitor 2
USP14 inhibitor
|
USP14-IN-2 is a specific small molecule USP14 inhibitor with IC50 of <0.5 uM. |
| PC-20186 |
USP14 inhibitor 1
USP14 inhibitor
|
USP14-IN-1 is a specific small molecule USP14 inhibitor with IC50 of 0.5 uM. |
| PC-20185 |
IU2-6
USP14 inhibitor
|
IU2-6 is a small molecule USP14 inhibitor, shows 74% inhibition at 8 uM. |
| PC-20184 |
GSK2643943A
USP20 inhibitor
|
GSK2643943A is a specific, cell penetrant small molecule inhibitor of deubiquitinating enzyme USP20 with IC50 of 160 nM (USP20/Ub-Rho). |
| PC-20004 |
TG2-179-1
BAP1 inhibitor
|
TG2-179-1 is a potent, selective and covalently inhibitor of deubiquitinase (DUB) BRCA1-associated protein-1 (BAP1), covalently binds to the active site of BAP1 (Cys91), exhibits potent cytotoxic activity against colon cancer cells. |
