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Request The Product List ofPI3K PI3K

Cat. No.	Product Name	Information
PC-61741	ST-168 MEK/PI3K inhibitor	ST-168 is a novel potent, orally available MEK/PI3K bifunctional inhibitor with IC50 of 182, 69.2, 1482, 2293, and 41.7 nM for MEK1, PI3Kα, PI3Kβ, PI3Kγ, and PI3Kδ, respectively.
PC-61135	PI3Kβ/δ inhibitor 20a PI3Kβ/δ inhibitor	PI3Kβ/δ inhibitor 20a is a potent, highly selective PI3Kβ/δ inhibitor with IC50 of 7.8/5.3 nM respectively, with liitle to no activity on PI3Kα/γ (IC50=850/>10,000 nM).
PC-61127	PI3Kδ inhibitor 52	ZUN64390 is a potent, selective, and efficacious PI3Kδ inhibitor with IC50 of 1.7 nM, >100-fold selectivitity over PI3Kγ/α/β.
PC-60983	AMG511 PI3K inhibitor	AMG511 (AMG-511) potent, efficacious, and orally available pan class I PI3K inhibitor with Ki of 4/6/2/1 nM for PI3Kα/β/δ/γ, respectively.
PC-60567	Tenalisib p110δ/γ inhibitor	Tenalisib (RP6530) is a potent, selective, orally active p110δ/γ PI3K dual inhibitor with IC50 of 24.5 and 33.2 nM, respectively.
PC-60566	IPI-443 p110δ/γ inhibitor	A potent, selective, orally active p110δ/γ PI3K dual inhibitor with cellular IC50 of 0.29 and 7.1 nM, respectively.
PC-60565	IPI-3063 p110δ inhibitor	IPI-3063 is apotent, and selective p110δ PI3K inhibitor with IC50 of 0.1 nM in cell-based assays.
PC-60527	Parsaclisib PI3Kδ inhibitor	Parsaclisib (INCB050465) is a potent and highly selective PI3Kδ inhibitor with IC50 of < 1 nM (SPA).
PC-60447	LAS191954 PI3Kδ inhibitor	LAS191954 is a potent, selective, orally bioavailable PI3Kδ inhibitor with IC50 of 2.6 nM.
PC-60413	SF-1126	SF-1126 is a pan PI3K/BRD4 inhibitor, RGDS-conjugated LY294002 prodrug that exhibits increased solubility and binds to specific integrins.
PC-60392	SN32976 PI3K/mTOR inhibitor	SN32976 is a novel, potent and selective class I PI3K and mTOR inhibitor with IC50 of 15.1/461/110/134/194 nM for PI3Kα/PI3Kβ/PI3Kγ/PI3Kδ/mTOR, respectively.
PC-60391	BL-140 p110β inhibitor	BL-140 is a potent, specific p110β inhibitor with IC50 of 5.74 nM.

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