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Request The Product List ofPI3K PI3K

Cat. No.	Product Name	Information
PC-21948	PIK-108 p110β inhibitor	PIK-108 is a potent, selective and allosteric PI3K p110β inhibitor with IC50 of 57 nM, 45-fold selective over PI3Kα (IC50=2600 nM).
PC-21947	PI3Kα H1047R inhibitor 17 H1047R PI3Kα inhibitor	PI3Kα H1047R inhibitor 17 is a potent, selective H1047R PI3Kα mutant inhibitor with IC50 of 1 nM (inhibition of pAKT formation), without effect on PI3Kα WT.
PC-21944	GSK2636771 PI3Kβ inhibitor	GSK2636771 is a potent, selective and orally bioavailable inhibitor of PI3Kβ with Ki/IC50 of 0.89/5.2 nM, respectively.
PC-20451	PITCOIN2 PI3KC2α inhibitor	PITCOIN2 (LU-06-006) is a potent selective PI3KC2α inhibitor with IC50 of 126 nM, has selectivity against PI3KC2γ but shows micromolar activity on PI3KC2β.
PC-42943	TGR-1202 R-enantiomer	TGR-1202 R-enantiomer is is the less active enantiomer of TGR-1202 (Umbralisib), TGR-1202 is a potent, selective, orally available PI3Kδ inhibitor with IC50 of 22 nM..
PC-42881	PI3K-IN-1	PI3K-IN-1 is a potent inhibitor of PI3K, extracted from patent WO2012103524 A2 and WO2013147649 A2..
PC-42647	PI3Kγ inhibitor 1	A potent PI3Kγ inhibitor..

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