PI3Kδ-IN-7n |CAS:2088525-31-7 Probechem Biochemicals

Chemical Structure : PI3Kδ-IN-7n

CAS No.: 2088525-31-7

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PI3Kδ-IN-7n

货号: PC-62806Not For Human Use, Lab Use Only.

PI3Kδ-IN-7n is a highly potent and selective PI3Kδ inhibitor with IC50 of 0.9 nM, displays high selectivity (>1,500-fold) over PI3Kα, PI3Kβ, PI3Kγ (IC50>1.5 uM).

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5 mg	￥2280	In stock
10 mg	￥3780	In stock
25 mg	￥5880	In stock
100 mg		Get quote

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生物&药学活性

PI3Kδ-IN-7n is a highly potent and selective PI3Kδ inhibitor with IC50 of 0.9 nM, displays high selectivity (>1,500-fold) over PI3Kα, PI3Kβ, PI3Kγ (IC50>1.5 uM).
PI3Kδ-IN-7n shows reasonable pharmacokinetics with good bioavailability and moderate in vivo half-life.
PI3Kδ-IN-7n is one of the most selective PI3Kδ inhibitors published to date.

物理化学性质&存储条件

分子量	429.459
分子式	C23H20FN7O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(3-amino-6-(1-methyl-5-(1-phenylcyclopropyl)-1H-1,2,4-triazol-3-yl)pyrazin-2-yl)-2-fluorobenzamide

参考文献

1. Terstiege I, et al. Bioorg Med Chem Lett. 2017 Feb 1;27(3):679-687.

PI3Kδ-IN-7n

生物&药学活性

物理化学性质&存储条件

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PI3Kδ-IN-7n

生物&药学活性

物理化学性质&存储条件

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