| Cat. No. |
Product Name |
Information |
| PC-61864 |
PF-04958242
AMPAR PAM
|
PF-04958242 (Pesampator) is a novel potent, selctive, and orally-active AMPA receptor (AMPAR) positive allosteric modulator (PAM) with Ki of 170 nM, EC50 of 370 nM. |
| PN-30006 |
Isomangiferin
|
Isomangiferin is the major tetracyclic oxindole alkaloid components of Uncaira species, inhibits NMDA receptor with IC50 of 43.2 uM, also blocks calcium channel. |
| PC-61727 |
CP-465022
AMPAR antagonist
|
CP-465022 is a potent, selective, noncompetitive AMPA receptor (AMPAR) antagonist with IC50 of 36 nM. |
| PC-61726 |
Tulrampator
AMPAR PAM
|
Tulrampator (S 47445, CX 1632) is a potent, selective, positive allosteric modulator of AMPA receptor (AMPAR) with EC50 of 2.5-5.4 uM for different AMPA receptors subtypes (GluA1/2/4 flip and flop variants). |
| PC-61725 |
GYKI 52466 dihydrochloride
AMPAR antagonist
|
GYKI 52466 is a selective, non-competitive, orally active AMPA receptor (AMPAR) antagonist with IC50 of 10-20 uM against AMPA-induced responses. |
| PC-61724 |
LY-404187
AMPAR PAM
|
LY-404187 is a potent, selective, positive allosteric modulator of AMPA receptor (AMPAR) with EC50 of 1.3 uM. |
| PC-61723 |
Org 26576
AMPAR PAM
|
Org 26576 (MK 8777, SCH 900777) is a potent AMPA receptor (AMPAR) positive allosteric modulator EC50 of 8-16 uM in rat hippocampal primary cultured neurons. |
| PC-61722 |
LY-503430
AMPAR agonist
|
LY-503430 is a novel AMPA receptor (AMPAR) potentiator that selectively enhances glutamate-induced calcium influx into HEK293 cells transfected with human GLUA1, GLUA2, GLUA3, or GLUA4 AMPA receptors with EC50 of 0.1-4 uM. |
| PC-61721 |
IDRA-21
AMPAR PAM
|
IDRA-21 is a positive allosteric modulator of the AMPA receptor (AMPAR). |
| PC-61720 |
NBQX disodium
AMPAR antagonist
|
NBQX disodium is the water soluble disodium salt of NBQX, which is a potent, selective and competitive AMPA receptor (AMPAR) antagonist with IC50 of 0.15 uM. |
| PC-61719 |
NBQX
AMPAR antagonist
|
NBQX is a potent, selective and competitive AMPA receptor (AMPAR) antagonist with IC50 of 0.15 uM. |
| PC-61718 |
CNQX disodium
AMPAR antagonist
|
CNQX disodium (FG 9065 disodium) is the water soluble disodium salt of CNQX, which is a potent AMPA/kainate receptor antagonist with IC50 of 0.3/1.5 uM, respectively.. |
