| Cat. No. |
Product Name |
Information |
| PC-60389 |
UMB-32
BRD4 inhibitor
|
UMB-32 is a potent, selective inhibitor of BRD4 with Kd of 550 nM, cellular IC50 of 724 nM. |
| PC-60388 |
UMB-136
|
UMB-136 (UMB136) is a novel bromodomain BRD4 inhibitor that significantly induces HIV-1 reactivation. |
| PC-60307 |
GNE-207
CBP/p300 inhibitor
|
GNE-207 (GNE207) is a novel potent, selective, orally active CBP/p300 bromodomain with IC50 of 1.0 nM. |
| PC-60306 |
GNE-781
CBP/p300 inhibitor
|
GNE-781 (GNE781) is a potent, selective, non-CNS penetrant, orally active CBP/p300 bromodomain inhibitor with IC50 of 0.94/1.2 nM in TR-FRET assays. |
| PC-60305 |
GNE-272
CBP/EP300 inhibitor
|
GNE-272 (GNE272) potent and selective the bromodomains of CBP/EP300 inhibitor with IC50 of 0.02 and 0.03 uM for CBP and EP300, respectively. |
| PC-60199 |
Ischemin
CBP bromodomain inhibitor
|
Ischemin is a cell permeable CBP bromodomain inhibitor with Kd of 19 uM. |
| PC-60198 |
Ischemin sodium
CBP bromodomain inhibitor
|
Ischemin sodium is a cell permeable CBP bromodomain inhibitor with Kd of 19 uM. |
| PC-60104 |
HJB97
BET inhibitor
|
HJB-97 (HJB97) is a potent BET bromodomian inhibitor with IC50 of 3-7 nM for BRD2/3/4 BD1 and BD2. |
| PC-70031 |
PF-CBP1
CBP/p300 inhibitor
|
PF-CBP1 is a potent, highly selective CBP/p300 bromodomains inhibitor with IC50 of 125 nM and 363 nM, respectively. |
| PC-70026 |
CPI-268456
BRD4 inhibitor
|
CPI-268456 is a small molecule ligand of bromodomain-containing protein 4 (BRD4), binds to BRD4 with IC50 of 0.5 uM in cell-free assays. |
| PC-60022 |
BAY-850
ATAD2 inhibitor
|
BAY-850 (BAY 850, BAY850) is a potent, isoform selective, cellularly active ATAD2 bromodomain inhibitor with binding IC50 of 166 nM in TR-FRET assay. |
| PC-45582 |
I-BRD9
BRD9 inhibitor
|
I-BRD9 is the first selective cellular chemical probe inhibitor for BRD9 with pIC50 of 7.3. |
