XDM-CBP |CAS:2138461-99-9 Probechem Biochemicals

Chemical Structure : XDM-CBP

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XDM-CBP (XDM CBP)

货号: PC-61151Not For Human Use, Lab Use Only.

XDM-CBP is a highly potent and selective inhibitor of CBP/p300 bromodomain with Kd of 0.23/0.47 uM respectively, with high selectivity over all other BD families, including the BET family.

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生物&药学活性

XDM-CBP is a highly potent and selective inhibitor of CBP/p300 bromodomain with Kd of 0.23/0.47 uM respectively, with high selectivity over all other BD families, including the BET family.
XDM-CBP exhibits antiproliferative effect on numerous cancer cell lines, in particular malignant melanoma, breast cancer, and leukemia (HL-60 and MCF-7 cells GI50=1.3 and 4.2 uM, respectively).

物理化学性质&存储条件

分子量	366.417
分子式	C21H22N2O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-acetyl-N-((2,8-dihydroxynaphthalen-1-yl)methyl)-3-ethyl-5-methyl-1H-pyrrole-2-carboxamide

参考文献

1. Hügle M, et al. Angew Chem Int Ed Engl. 2017 Aug 2. doi: 10.1002/anie.201705516.

XDM-CBP (XDM CBP)

生物&药学活性

物理化学性质&存储条件

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XDM-CBP (XDM CBP)

生物&药学活性

物理化学性质&存储条件

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