| Cat. No. |
Product Name |
Information |
| PC-61562 |
APD916
Histamine H3 antagonist
|
APD916 is a potent and selective antagonist of the H3 receptor with Ki of 0.7 nM for rH3R. |
| PC-61337 |
MK-7288
H3R inverse agonist
|
MK-7288 is a selective histamine H3 receptor inverse agonist for the treatment of sleep apnoea syndrome. |
| PC-60793 |
JNJ-39758979
Histamine H4 antagonist
|
JNJ-39758979 (JNJ39758979) is a potent, selective, orally bioavailable histamine H4 receptor (H4R) antagonist with Ki of 12.5 nM, >80-fold selectivity over other histamine receptors. |
| PC-60533 |
Seliforant
Histamine H4 antagonist
|
Seliforant (SENS-111, SENS111) is a novel potent, selective histamine H4 receptor antagonist. |
| PC-60377 |
S 38093
Histamine H3 antagonist
|
S 38093 is a brain-penetrant H3 receptor antagonist/inverse agonist that shows procognitive properties in vivo. |
| PC-45168 |
Loratadine
Histamine H1 agonist
|
A tricyclic antihistamine that acts as a selective inverse agonist of peripheral histamine H1-receptors.. |
| PC-45167 |
Cetirizine dihydrochloride
Histamine H1 antagonist
|
Cetirizine dihydrochloride is a second-generation antihistamine that acts as a selective H1 receptor antagonist, inhibits eosinophil chemotaxis during the allergic response. |
| PC-45166 |
Cetirizine
Histamine H1 antagonist
|
Cetirizine is a second-generation antihistamine that acts as a selective H1 receptor antagonist, inhibits eosinophil chemotaxis during the allergic response. |
| PC-42380 |
VUF10460
Histamine H4 agonist
|
VUF10460 is a potent, selective histamine H4 receptor (H4R) agonist with pKi of 7.46 and 8.22 for rat and human H4, respectively. |
| PC-45369 |
Decloxizine
Histamin H1 antagonist
|
Decloxizine (UCB-1402, NSC-289116) is a potent histamine 1 (H1) receptor antagonist. |
| PC-42908 |
ABT-239
Histamine H3 antagonist
|
ABT-239 is a potent and selective Histamine H3 receptor antagonist with Ki of 0.1-5.8 nM (human, rat H3). |
| PC-42911 |
Pitolisant hydrochloride
H3 receptor antagonist
|
Pitolisant hydrochloride (Ciproxidine, BF2649) is a potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM. |
