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首页-小分子抑制剂&激动剂-GPCR-Histamine Receptor-VUF10460
VUF10460

Chemical Structure : VUF10460

CAS No.: 1028327-66-3

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VUF10460 (VUF-10460, VUF 10460)

货号: PC-42380Not For Human Use, Lab Use Only.

VUF10460 is a potent, selective histamine H4 receptor agonist with pKi of 7.46 and 8.22 for rat and human H4, respectively.

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5 mg ￥880 In stock
10 mg ￥1280 In stock
25 mg ￥2180 In stock
50 mg ￥3580 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

VUF10460 is a potent, selective histamine H4 receptor agonist with pKi of 7.46 and 8.22 for rat and human H4, respectively.
VUF10460 displays >50-fold selectivity over H3 receptors.
VUF10460 significantly enhances HCl-induced gastric lesions in rat stomach, but not the H3 selective agonist JNJ7777120.

物理化学性质&存储条件

分子量 269.34486
分子式 C15H19N5
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

DMSO: ≥ 36 mg/mL
Chemical Name/SMILES

2-Pyrimidinamine, 4-(4-methyl-1-piperazinyl)-6-phenyl-

参考文献

1. Coruzzi G, et al. Eur J Pharmacol. 2011 Nov 1;669(1-3):121-7.

2. Adami M, et al. Pharmacology. 2012;89(5-6):287-94.

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