欢迎访问ProbeChem中文网站，英文网站请访问www.probechem.com
    英文 |     中文

产品咨询: sales@probechem.com
订购: order@probechem.com

首页-小分子抑制剂&激动剂-GPCR-Histamine Receptor-ABT-239
ABT-239

Chemical Structure : ABT-239

CAS No.: 460746-46-7

加入收藏

ABT-239 (ABT239, ABT 239)

货号: PC-42908Not For Human Use, Lab Use Only.

ABT-239 is a potent and selective Histamine H3 receptor antagonist with Ki of 0.1-5.8 nM (human, rat H3).

规格 价格 库存 数量
5 mg ￥980 In stock
10 mg ￥1580 In stock
25 mg ￥2780 In stock
50 mg ￥4780 In stock
100 mg Get quote
获取报价单
* 请选择数量再加入购物车
 or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

ABT-239 is a potent and selective Histamine H3 receptor antagonist with Ki of 0.1-5.8 nM (human, rat H3).
ABT-239 exhibits 1000-fold selectivity versus H1, H2 and H4.
ABT-239 exhibits excellent pharmacokinetic and metabolic properties across species and good oral bioavailability.

物理化学性质&存储条件

分子量 330.4229
分子式 C22H22N2O
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

DMSO: ≥ 3.3 mg/mL
Chemical Name/SMILES

Benzonitrile, 4-[2-[2-[(2R)-2-methyl-1-pyrrolidinyl]ethyl]-5-benzofuranyl]-

参考文献

1. Cowart M, et al. J Med Chem. 2005 Jan 13;48(1):38-55.

2. Esbenshade TA, et al. J Pharmacol Exp Ther. 2005 Apr;313(1):165-75.

3. Bhowmik M, et al. Brain Res. 2014 Sep 18;1581:129-40.

备案号：沪ICP备16042516号-1 Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

联系我们 sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

询单

  • *产品名称:
  • *姓名:
  • *邮箱:
  • *公司名称:
  • *询单数量:
  • *国籍:
  • 询单信息: