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首页-小分子抑制剂&激动剂-GPCR-Histamine Receptor-APD916
APD916

Chemical Structure : APD916

CAS No.: 1021169-11-8

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APD916 (APD-916)

货号: PC-61562Not For Human Use, Lab Use Only.

APD916 is a potent and selective antagonist of the H3 receptor with Ki of 0.7 nM for rH3R.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    APD916 is a potent and selective antagonist of the H3 receptor with Ki of 0.7 nM for rH3R.
    APD916 increases wakefulness in rodents as measured by polysomnography with a duration of effect consistent with its pharmacokinetic properties.

    物理化学性质&存储条件

    分子量 401.565
    分子式 C23H31NO3S
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (R)-1-(2-(4'-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl)-2-methylpyrrolidine

    参考文献

    1. Semple G, et al. Bioorg Med Chem Lett. 2012 Jan 1;22(1):71-5.

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