| Cat. No. |
Product Name |
Information |
| PC-49736 |
UR-Po563
H2 receptor agonist
|
UR-Po563 is a potent, selective H2 receptor agonist with pKi of 7.75, >400-fold selectivity over H1R/H3R/H4R. |
| PC-47094 |
RGH-235
H3R antagonist
|
RGH-235 is a potent, selective, and orally active H3 receptor antagonist/inverse agonist with high affinity (Ki=3.0-9.2 nM, depending on species), without affinity to H1, H2 or H4 receptors. |
| PC-72278 |
TASP0410461
H3R antagonist
|
TASP0410461 is a potent, selective histamine H3 receptor antagonist/inverse agonist. |
| PC-72277 |
Enerisant hydrochloride
H3R antagonist
|
Enerisant hydrochloride (TS091 hydrochloride) is a potent, selective histamine H3 receptor antagonist/inverse agonist with IC50 of 2.89 and 14.5 nM against hH3R and rH3R, respectively. |
| PC-72276 |
Enerisant
H3R antagonist
|
Enerisant (TS091,TS-091) is a potent, selective histamine H3 receptor antagonist/inverse agonist with IC50 of 2.89 and 14.5 nM against hH3R and rH3R, respectively. |
| PC-36072 |
VUF15000
Histamine H3 agonist
|
VUF15000 (VUF-15000) is the first photoswitchable GPCR Histamine H3 receptor agonist (pKi=8.42), displays >300-fold selective for hH3R over hH1R and hH2R. |
| PC-36071 |
NLX-204
5-HT1A agonist
|
NLX-204 (NLX204) is a potent, selective, ERK1/2 phosphorylation-preferring serotonin 5-HT1A receptor agonist with pEC50 of 9.37. |
| PC-36027 |
K-8986 maleate
Histamine H1 antagonist
|
K-8986 maleate (K8986) is a histamine H1-receptor antagonist with potential therapeutic for treatment of allergic conjunctivitis. |
| PC-35982 |
SUVN-G3031 free base
H3R inverse agonist
|
SUVN-G3031 (Samelisant) free base is a potent, selective, orally active histamine H3 receptor (H3R) inverse agonist with Ki of 8.73 nM (hH3R). |
| PC-35981 |
SUVN-G3031
H3R inverse agonist
|
SUVN-G3031 (Samelisant) is a potent, selective, orally active histamine H3 receptor (H3R) inverse agonist with Ki of 8.73 nM (hH3R). |
| PC-35408 |
JNJ-5207852
H3R antagonist
|
JNJ-5207852 (JNJ5207852) is a potent, selective antagonist of H3 receptor with pKi of 8.9 and 9.24 for rat and human H3, respectively. |
| PC-35407 |
Contilisant
AChE inhibitor
|
Contilisant is a neuroprotective, non-toxic, antioxidant, permeable ligand, showing in vitro pharmacological properties on the selected biological targets (hAChE IC50=0.53 uM. |
