UR-Po563 | H2 receptor agonist | Probechem Biochemicals

Chemical Structure : UR-Po563

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UR-Po563 (UR-Po 563)

货号: PC-49736Not For Human Use, Lab Use Only.

UR-Po563 is a potent, selective H2 receptor agonist with pKi of 7.75, >400-fold selectivity over H1R/H3R/H4R.

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生物&药学活性

UR-Po563 is a potent, selective H2 receptor agonist with pKi of 7.75, >400-fold selectivity over H1R/H3R/H4R.
UR-Po563 increased force of contraction in left atrium from H2-TG mice with pEC50 values of 8.27.
UR-Po563 increased force of contraction in isolated human right atrial muscle strips.

物理化学性质&存储条件

分子量	360.48
分子式	C17H24N6OS
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Urea, N-[[[3-(2-amino-4-methyl-5-thiazolyl)propyl]amino]iminomethyl]-N′-[(1R)-1-phenylethyl]-

参考文献

1. Ulrich Gergs, et al. J Pharmacol Exp Ther. 2021 Nov;379(3):223-234.

2. Biselli S, et al. Eur J Med Chem 214:113190

UR-Po563 (UR-Po 563)

生物&药学活性

物理化学性质&存储条件

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UR-Po563 (UR-Po 563)

生物&药学活性

物理化学性质&存储条件

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