Pitolisant hydrochloride (Ciproxidine) | H3 receptor antagonist

Chemical Structure : Pitolisant hydrochloride

CAS No.: 903576-44-3

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Pitolisant hydrochloride (Ciproxidine, BF2649, BF-2649)

货号: PC-42911Not For Human Use, Lab Use Only.

Pitolisant hydrochloride (Ciproxidine, BF2649) is a potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.

规格	价格	库存
10 mg	￥780	In stock
25 mg	￥1280	In stock
50 mg	￥2180	In stock
100 mg	￥3580	In stock
250 mg		Get quote

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生物&药学活性

Pitolisant hydrochloride (Ciproxidine, BF2649) is a potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.
Pitolisant hydrochloride has no effect on H1, H2, H4 receptors (IC50>10 uM); orally bioactive.

物理化学性质&存储条件

分子量	332.3084
分子式	C17H27Cl2NO
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: ≥ 43 mg/mL
Chemical Name/SMILES	Piperidine, 1-[3-[3-(4-chlorophenyl)propoxy]propyl]-, hydrochloride (1:1)

参考文献

1. Ligneau X, et al. J Pharmacol Exp Ther. 2007 Jan;320(1):365-75.

2. Dudek M, et al. Metab Brain Dis. 2016 Oct;31(5):1023-9.

3. Ligneau X, et al. Biochem Pharmacol. 2007 Apr 15;73(8):1215-24.

Pitolisant hydrochloride (Ciproxidine, BF2649, BF-2649)

生物&药学活性

物理化学性质&存储条件

参考文献

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Pitolisant hydrochloride (Ciproxidine, BF2649, BF-2649)

生物&药学活性

物理化学性质&存储条件

参考文献

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