| Cat. No. |
Product Name |
Information |
| PC-63551 |
Zicronapine
|
Zicronapine (Lu 31-130) is an antipsychotic agent that shows potent antagonistic effects at dopamine D1, D2 and serotonin 5HT2A receptors, exhibits monoaminergic activity and has a multi-receptorial profile. |
| PC-63550 |
BL-1020
|
BL-1020 is an ester of GABA and perphenazine, fuctions as orally-active antipsychotic agent and acts as a D2 antagonist and GABA agonist. |
| PC-63349 |
BRD5814
D2R inhibitor
|
BRD5814 is a potent, selective, highly brain penetrant β-arrestin biased dopamine D2 receptor (D2R) antagonist with Ki of 0.27 uM. |
| PC-43160 |
Bromocriptine mesylate
D2R agonist
|
Bromocriptine (CB-154) is a dopamine D2 receptor agonist (Ki=3 nM) and and various serotonin receptors, also inhibits the release of glutamate by reversing the glutamate GLT1 transporter. |
| PC-42975 |
SB269652
D2R/D3R modulator
|
SB269652 is a potent, selective, negative allosteric modulator of dopamine D2 and D3 receptors, abolishes specific binding of [3H]nemanopride and [3H]spiperone to CHO-transfected D3 receptors with IC50 of1.86 and 0.18 nM. |
| PC-63187 |
Brilaroxazine
Dopamine/5-HT modulator
|
RP-5063 (Brilaroxazine) is a multimodal dopamine and serotonin modulator with partial agonist activity at DA D2, D3, D4, 5-HT1A, and 5-HT2ARs, and antagonist activity at 5-HT2B, 5-HT6 and 5-HT7Rs. |
| PC-63113 |
A-68930 hydrochloride
D1DR agonist
|
A-68930 is a potent, specific, orally bioavailable agonist of the D1 dopamine receptor (D1DR) with EC50 of 2.5 nM. |
| PC-62128 |
ML398
D4R inhibitor
|
ML398 (CID72737723) is a potent, selective, highly brain penetrant dopamine 4 (D4R) receptor antagonist with IC50/Ki of 130 nM/60 nM. |
| PC-61749 |
Alizapride hydrochloride
D2R antagonist
|
Alizapride (MS 5080) is a dopamine D2 antagonist with prokinetic and antiemetic effects used in the treatment of nausea and vomiting.. |
| PC-61748 |
Alizapride
D2R antagonist
|
Alizapride (MS 5080) is a dopamine D2 antagonist with prokinetic and antiemetic effects used in the treatment of nausea and vomiting. |
| PC-61736 |
BP 897
D3R agonist
|
BP 897 is the first, potent, selective partial dopamine D3 receptor agonist with Ki of 0.92 nM. |
| PC-61553 |
JNJ-37822681
D2R antagonist
|
JNJ-37822681 is a potent, specific and fast-dissociating dopamine D2 antagonist with Ki of 158 nM. |
