| Cat. No. |
Product Name |
Information |
| PC-42584 |
SKF-82958 hydrobromide
Dopamine D1 agonist, ERα agonist
|
SKF-82958 hydrobromide is a potent, full dopamine D1 agonist, produces characteristic anorectic effects, hyperactivity and self-administration in animals. |
| PC-42583 |
SKF 82958
Dopamine D1 agonist, ERα agonist
|
SKF 82958 is a potent, full dopamine D1 agonist, produces characteristic anorectic effects, hyperactivity and self-administration in animals. |
| PC-45204 |
Metoclopramide
D2R antagonist
|
Metoclopramide is apotent dopamine D2 receptor antagonist with Ki of 28 nM. |
| PC-42716 |
SB-277011
D3R antagonist
|
SB-277011 (SB277011A) is a potent and selective dopamine D3 receptor antagonist with pKi of 8.0. |
| PC-46554 |
Pramipexole
Dopamine receptor agonist
|
Pramipexole is a partial/full agonist of dopamine receptor with Ki of 3.9/2.2/0.5/5.1 nM for D2S/D2L/D3/D4 respectively, also possesses low/insignificant affinity (500-10,000 nM) for the 5-HT1A, 5-HT1B, 5-HT1D, and α2-adrenergic receptors. |
| PC-45175 |
Dexpramipexole
Dopamine receptor agonist
|
Dexpramipexole ((R)-Pramipexole) is a partial/full agonist of dopamine receptor with Ki of 3.9/2.2/0.5/5.1 nM for D2S/D2L/D3/D4, respeectively. |
| PC-45174 |
Dexpramipexole dihydrochloride
Dopamine receptor agonist
|
Dexpramipexole dihydrochloride ((R)-Pramipexole) is a partial/full agonist of dopamine receptor with Ki of 3.9/2.2/0.5/5.1 nM for D2S/D2L/D3/D4, respeectively. |
| PC-45173 |
Pramipexole dihydrochloride
Dopamine receptor agonist
|
Pramipexole dihydrochloride is a partial/full agonist of dopamine receptor with Ki of 3.9/2.2/0.5/5.1 nM for D2S/D2L/D3/D4, respeectively. |
| PC-26861 |
PG01037 dihydrochloride
D3R antagonist
|
PG01037 dihydrochloride is a potent selective dopamine D3 receptor (D3R) antagonist with binding Ki of 0.7 nM, displays 133- and 540-fold selectivity over D2 and D4 receptors, respectively. |
| PC-26860 |
PG01042
D3R agonist
|
PG01042 is a high affinity, selective D3 dopamine receptor (D3R) agonist with Ki of 0.47 nM, 39-fold selective over D2R. |
| PC-26137 |
ENX-104
D2/D3 receptor antagonist
|
ENX-104 is a highly selective and potent dopamine D2/D3 receptor antagonist with IC50 of 1.1 nM, 0.1 nM, 2.4 nM and 15.3 nM for D2-like inhibitory dopamine receptors D2S, D2L, D3, and D4 respectively. |
| PC-26129 |
Thioridazine
D2R antagonist
|
Thioridazine is a selective antagonist of dopamine receptor D2 family proteins, exhibits potent anti-psychotic and anti-anxiety activities. |
