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首页-小分子抑制剂&激动剂-GPCR-Dopamine Receptor-PF-219061
PF-219061

Chemical Structure : PF-219061

CAS No.: 710654-74-3

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PF-219061 (PF 219061, PF219061)

货号: PC-70057Not For Human Use, Lab Use Only.

PF-219061 (PF 219061, PF219061) is a potent, selective agonist of dopamine D3 receptor with EC50 of 8 nM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    PF-219061 (PF 219061, PF219061) is a potent, selective agonist of dopamine D3 receptor with EC50 of 8 nM.
    PF-219061 has >1000-fold functional selectivity over D2, displays minimal binding activity (IC50>10 uM) against a wide panel of targets including dopamine D1 and D5 receptors.
    PF-219061 demonstrates activity in animal models of male erectile dysfunction.

    物理化学性质&存储条件

    分子量 235.327
    分子式 C14H21NO2
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    3-((2R,5S)-5-methyl-4-propylmorpholin-2-yl)phenol

    参考文献

    1. Blagg J, et al. Bioorg Med Chem Lett. 2007 Dec 15;17(24):6691-6.

    2. Attkins NJ, et al. Xenobiotica. 2009 Jul;39(7):523-33.

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