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首页-小分子抑制剂&激动剂-GPCR-Dopamine Receptor-PF-06256142
PF-06256142

Chemical Structure : PF-06256142

CAS No.: 1609583-14-3

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PF-06256142 (PF06256142)

货号: PC-35799Not For Human Use, Lab Use Only.

PF-06256142 (PF06256142) is a potent and selective orthosteric agonist of the D1 receptor with EC50 (cAMP) of 33 nM, shows exquisitely selectivity over D2.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    PF-06256142 (PF06256142) is a potent and selective orthosteric agonist of the D1 receptor with EC50 (cAMP) of 33 nM, shows exquisitely selectivity over D2.
    PF-06256142 demonsrates reduced receptor desensitization relative to dopamine and other catechol-containing agonists.

    物理化学性质&存储条件

    分子量 356.385
    分子式 C21H16N4O2
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (+)-4-(3-Methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)phenoxy)furo[3,2-c]pyridine

    参考文献

    1. Davoren JE, et al. J Med Chem. 2018 Nov 15. doi: 10.1021/acs.jmedchem.8b01622.

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