| Cat. No. |
Product Name |
Information |
| PC-35627 |
BTX-A51
CK1α inhibitor, CDK7/9 inhibitor
|
BTX-A51 (CK1α inhibitor A51) is a novel pan-specific CK1 (CSNK1) inhibitor (Kd=0.5-20 nM, CK1α Kd=5.3 nM) that co-targets the transcriptional kinases CDK7 and CDK9, with hardly inhibition of CDK8, CDK13, CDK11a, CDK11b, and CDK19. |
| PC-35616 |
BMS-699
CK2 inhibitor
|
BMS-699 (BMS699) is a novel potent, selective, ATP-competitive casein kinase 2 (CK2) inhibitor with IC50 of 0.1 nM (CKα). |
| PC-35185 |
CAM4712
CK2α inhibitor
|
CAM4712 (CAM-4712) is a potent and selective CK2alpha (CK2α) inhibitor with IC50 of 7 uM, exhibits cell growth inhibition in HCT116 cell line with IC50 of 10 uM. |
| PC-35184 |
CAM4066
CK2α inhibitor
|
CAM4066 (CAM-4066) is a potent and selective CK2alpha (CK2α) inhibitor with Kd of 0.32 uM and IC50 of 0.37 uM, shows significantly improved selectivity compared to other CK2α inhibitors. |
| PC-43200 |
IC261
CK1δ/CK1ε inhibitor
|
IC261 (IC-261, SU-5607) is a potent, specific, ATP-competitive CK1delta/epsilon (CK1δ/CK1ε) with IC50 of 1 uM, does not block the activity of α, β and γ isoforms. |
| PC-62834 |
CK1-IN-3c
CK1δ/ε inhibitor
|
CK1-IN-3c is a novel casein kinase 1δ/ε (CK1δ/ε) inhibitor with IC50 of 1.6 uM. |
| PC-62346 |
CK2-IN-1
CK2 inhibitor
|
CK2-IN-1 is a potent, competitive inhibitor of ATP binding to Casein kinase 2 (CK2) with IC50 of 9 nM, induces differentiation of epidermal progenitor cells to terminally differentiated keratinocytes with EC50 of 0.1 uM. |
| PC-62192 |
Quinalizarin
CK2 inhibitor
|
Quinalizarin is a potent, selective and cell-permeable inhibitor of CK2 with Ki of 58 nM. |
| PC-61326 |
TBBz
CK2 inhibitor
|
TBBz is a potent, selective and ATP-competitive CK2 inhibitor with Ki of 0.5-1 uM. |
| PC-61114 |
PF-5006739
CK1δ/ε inhibitor
|
PF-5006739 is a potent, selective casein kinase CK1δ/ε inhibitor with IC50 of 3.9/17.0 nM, respectively. |
| PC-60582 |
(R)-DRF053 dihydrochloride
CK1/CDK inhibitor
|
(R)-DRF053 dihydrochloride (DRF053) is a potent, cell-permeable, dual CK1/CDK inhibitor with IC50 of 14 nM, 220 nM and 80 nM for CK1, CDK5/p25 and CDK1/cyclin B, respectively. |
| PC-60581 |
Bischof-5
CK1δ inhibitor
|
Bischof-5 (CK1δ inhibitor 5) is a potent, specific casein kinase 1δ (CK1δ) inhibitor with IC50 of 40 nM. |
