P-glycoprotein (P-gp) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofP-glycoprotein (P-gp) P-glycoprotein (P-gp)

Cat. No.	Product Name	Information
PC-20572	Ceefourin-1 MRP4/ABCC4 inhibitor	Ceefourin-1 is a highly selective inhibitor of multidrug resistance protein 4 (MRP4/ABCC4), inhibits the efflux of a broad range of MRP4 substrates.
PC-73219	Encequidar mesylate monohydrate MDR1 inhibitor	Encequidar (HM30181) mesylate monohydrate is a potent selective inhibitor of MDR1 (ABCB1, P-gp) with IC50 of 0.63 nM.
PC-73218	Encequidar MDR1 inhibitor	Encequidar (HM30181) is a potent selective inhibitor of MDR1 (ABCB1, P-gp) with IC50 of 0.63 nM.
PC-72608	CP-100356 hydrochloride P-gp inhibitor	CP-100356 hydrochloride (CP100356) is a specific P-glycoprotein (P-gp) inhibitor, suppresses VSV-LASVGP, LCMV, and LASV infection with IC50 of 0.52, 0.54, and 0.062 uM, respectively, without significant cytotoxicity.
PC-62666	NSC23925B P-gp inhibitor	NSC23925B is a small molecule agent that reverses MDR in cancer cells, reverses MDR in several drug-resistant cell lines expressing P-gp.
PC-62665	NSC23925 P-gp inhibitor	NSC 23925 is a small molecule compound that reverses multiple drug resistance (MDR) in human cancer cell lines, reverses MDR1 (Pgp1) but does not inhibit MRP or BCRP-mediated MDR.
PC-70022	Laniquidar P-gp inhibitor	Laniquidar (R101933) is an orally active, third-generation P-glycoprotein inhibitor that inhibits the drug efflux pump P-glycoprotein, resulting in higher concentrations of antineoplastic agents in tumor cells that are multi-drug resistant due to the overexpression of P-glycoprotein.
PC-42648	Tariquidar P-gp inhibitor	Tariquidar (XR9576) is a potent, specific P-gp inhibitor with Kd of 5.1 nM.
PC-45836	Zosuquidar trihydrochloride P-gp inhibitor	Zosuquidar trihydrochloride (LY335979) is a potent P-glycoprotein (P-gp) inhibitor with Ki of 60 nM.
PC-45888	Elacridar hydrochloride P-gp inhibitor	Elacridar hydrochloride is a potent inhibitor of multidrug resistance (MDR, P-gp) that fully reverses multidrug resistance CHRC5, OV1/DXR and MCF7/ADR cells to the cytotoxicity of doxorubicin and vincristine with IC50 of 0.02 uM.
PC-45887	Elacridar P-gp inhibitor	Elacridar (GF120918, GW-0918) is a potent inhibitor of multidrug resistance (MDR, P-gp) that fully reverses multidrug resistance CHRC5, OV1/DXR and MCF7/ADR cells to the cytotoxicity of doxorubicin and vincristine with IC50 of 0.02 uM.
PC-45137	Dofequidar fumarate P-gp inhibitor	Dofequidar fumarate (MS-209) is an orally active quinoline compound that can reverse P-glycoprotein (P-gp)-mediated MDR.

PREV12 NEXT