Laniquidar | P-gp inhibitor | Probechem Biochemicals

Chemical Structure : Laniquidar

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Laniquidar (R-101933, R101933)

货号: PC-70022Not For Human Use, Lab Use Only.

Laniquidar (R101933) is an orally active, third-generation P-glycoprotein inhibitor that inhibits the drug efflux pump P-glycoprotein, resulting in higher concentrations of antineoplastic agents in tumor cells that are multi-drug resistant due to the overexpression of P-glycoprotein.

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生物&药学活性

Laniquidar (R101933) is an orally active, third-generation P-glycoprotein (P-gp) inhibitor that inhibits the drug efflux pump P-glycoprotein, resulting in higher concentrations of antineoplastic agents in tumor cells that are multi-drug resistant due to the overexpression of P-glycoprotein.

物理化学性质&存储条件

分子量	584.7
分子式	C37H36N4O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	methyl 11-(1-(4-(quinolin-2-ylmethoxy)phenethyl)piperidin-4-ylidene)-6,11-dihydro-5H-benzo[d]imidazo[1,2-a]azepine-3-carboxylate

参考文献

1. van Zuylen L, et al. Clin Cancer Res. 2000 Apr;6(4):1365-71.

2. van Zuylen L, et al. Eur J Cancer. 2002 May;38(8):1090-9.

3. Luurtsema G, et al. Nucl Med Biol. 2009 Aug;36(6):643-9.

Laniquidar (R-101933, R101933)

生物&药学活性

物理化学性质&存储条件

参考文献

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Laniquidar (R-101933, R101933)

生物&药学活性

物理化学性质&存储条件

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