Ribosomal S6 Kinase (RSK) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofRibosomal S6 Kinase (RSK) Ribosomal S6 Kinase (RSK)

Cat. No.	Product Name	Information
PC-21764	BIX 02565 RSK2 inhibitor	BIX 02565 is a potent, selective ribosomal S6 kinase 2 (RSK2) inhibitor with IC50 of 1.1 nM.
PC-49024	PF-4708671 S6K1 inhibitor	PF-4708671 is a potent, specific, cell-permeable inhibitor of S6K1 (p70 ribosomal S6 kinase 1), inhibits the activity of full-length S6K1 in vitro with Ki of 20 nM, and S6K1 isolated from IGF1-stimulated HEK293 cells with IC50 of 160 nM.
PC-72701	S6K2 inhibitor Compound 2 S6K2 inhibitor	S6K2 inhibitor Compound 2 is the first potent and highly isoform-specific S6K2 inhibitor with IC50 of 22 nM, inactive for the closely related isoform S6K1 at 5 uM.
PC-72284	PMD-026 RSK inhibitor	PMD-026 (PMD026) is an oral, reversible small molecule inhibitor of ribosomal S6 kinases (RSK1-4) with IC50 of 2 nM (RSK1), 0.7 nM (RSK2), 0.9 nM (RSK3) and 2 nM (RSK4).
PC-43060	LY-2584702 hydrochloride p70S6K1 inhibitor	LY2584702 is a potent, selective, ATP-competitive inhibitor of P70S6 kinase-1 (p70S6K1) with IC50 of 4 nM.
PC-43059	LY-2584702 tosylate p70S6K1 inhibitor	LY-2779964 (LY2584702 tosylate) is a potent, selective, ATP-competitive inhibitor of P70 S6 kinase-1 (p70S6K1) with IC50 of 4 nM.
PC-43058	LY-2584702 p70S6K1 inhibitor	LY2584702 is a potent, selective, ATP-competitive inhibitor of P70 S6 kinase-1 (p70S6K1) with IC50 of 4 nM.
PC-62854	RSK2-IN-20 RSK2 inhibitor	RSK2-IN-20 is a potent, selective, and durable inhibitpr of RSK2 with IC50 of 47 nM.
PC-62045	BRD 7389 RSK inhibitor	BRD 7389 is an inhibitor of ribosomal S6 kinases (RSK) with IC50 of 1.5 uM, 2.4 uM, and 1.2 uM for RSK1, RSK2, and RSK3, respectively.
PC-60433	M2698 S6K/Akt inhibitor	M2698 (MSC2363318A) is a potent, selective, ATP-competitive, orally bioavailable and brain penetrant dual inhibitor of p70S6K and Akt1/3 with IC50 of 1 nM and 17 nM, respectively.
PC-70183	SL0101 RSK inhibitor	SL0101 (SL 0101-1) is the first specific inhibitor of RSK (p90 ribosomal S6 kinase) with IC50 of 89 nM for RSK2.
PC-45678	LJI308 RSK inhibitor	LJI308 (LJI 308) is a potent and specific pan-RSK inhibitor with IC50s of 6 nM, 4 nM and 13 nM for RSK1, RSK2 and RSK3 respectively.

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