| Cat. No. |
Product Name |
Information |
| PC-62558 |
Garcinol
p300/PCAF inhibitor
|
Garcinol (Camboginol) is a potent, natural inhibitor of histone acetyltransferases (HATs) p300 (IC50=7 uM) and PCAF (IC50=5 uM) both in vitro and in vivo. |
| PC-62267 |
SPV106
p300/PCAF activator
|
SPV 106 is the first mixed activator/inhibitor of Histone acetyltransferases (HATs), potentiates p300/CBP-associated factor (PCAF) HAT activity while inhibiting those of p300/CBP and recombinant CBP. |
| PC-62266 |
CTPB
p300 activator
|
CTPB is an anacardic acid derivative, was reported as a selective activator of p300 (KAT3B) HAT activity but not PCAF (KAT2B), which enhanced HAT-dependent transcriptional activation. |
| PC-61762 |
L-002
KAT3B inhibitor
|
L-002 (NSC 764414, L002) is a novel potent, specific acetyltransferase p300 (KAT3B) inhibitor with IC50 of 1.98 uM. |
| PC-61686 |
PU-139
HAT inhibitor
|
PU-139 is a potent, unselective HAT (Histone acetyltransferase) inhibitor that blocks the HATs Gcn5, p300/CBP-associated factor (PCAF), CREB protein (CBP) and p300. |
| PC-61685 |
PU-141
p300/CBP inhibitor
|
PU-141 is a potent, selective CBP/p300 inhibitor that inhibits SK-N-SH cell growth with GI50 of 0.48 uM. |
| PC-60499 |
TH1834 dihydrochloride
Tip60 inhibitor
|
TH1834 dihydrochloride (TH-1834, TH 1834) is a novel potent specific histone acetyltransferase Tip60 inhibitor. |
| PC-60498 |
TH1834
Tip60 inhibitor
|
TH1834 (TH-1834, TH 1834) is a novel potent specific histone acetyltransferase Tip60 inhibitor. |
| PC-70121 |
Windorphen
p300 inhibitor
|
Windorphen is a potent, selective inhibitor of p300 histone acetyltransferase (IC50=4.2 uM). |
| PC-60028 |
A-485
p300/CBP inhibitor
|
A-485 (A485) is a potent, selective and, cell and in vivo active p300/CBP catalytic inhibitor with IC50 of 9.8/2.6 nM. |
| PC-45646 |
I-CBP112
CBP/p300 inhibitor
|
I-CBP112 is a specific and potent inhibitor of CBP/p300 bromodomain with Kd of 150-170 nM. |
| PC-45052 |
Remodelin hydrobromide
NAT10 inhibitor
|
Remodelin hydrobromide is a potent inhibitor of the acetyl-transferase protein NAT10 that acetylates both histones and microtubules. |
