| Cat. No. |
Product Name |
Information |
| PC-45051 |
Remodelin
NAT10 inhibitor
|
Remodelin is a potent inhibitor of the acetyl-transferase protein NAT10 that acetylates both histones and microtubules. |
| PC-24171 |
Prifetrastat
KAT6A/6B inhibitor
|
Prifetrastat (PF-07248144) is a potent, selective histone acetyltransferase KAT6 (KAT6A/6B) inhibitor. |
| PC-24033 |
EPS496
p300 inhibitor
|
EPS496 is a small molecule inhibitor of histone acetyltransferase p300, binds effectively to p300 and inhibits p300 kinase activation. |
| PC-23724 |
CHI-KAT8i5
KAT8 inhibitor
|
CHI-KAT8i5 is a specific small molecule inhibitor of KAT8 (lysine acetyltransferase 8), directly binds to KAT8 with SPR KD of 19.72 uM, suppresses esophageal squamous cell carcinoma (ESCC) growth through targeting KAT8/c-Myc signaling pathway. |
| PC-21986 |
EPIC-0628
HOTAIR-EZH2 inhibitor
|
EPIC-0628 (EPIC0628) is a selective and potent inhibitor that selectively disrupts the HOTAIR-EZH2 interaction and promotes ATF3 expression, enhances the temozolomide efficacy in glioblastoma. |
| PC-21843 |
SGF29 inhibitor DC60
SGF29 inhibitor
|
SGF29 inhibitor DC60 is a small molecule inhibitor of Spt-Ada-Gcn5 acetyltransferase (SAGA)-associated factor 29 (SGF29, CCDC101) with IC50 of 6.4 uM, binds to SGF29 second Tudor domain (SGF29 Tudor 2) and blocks SGF29 chromatin binding domain. |
| PC-20867 |
MG149
Tip60 (KAT5) inhibitor
|
MG149 is a selective histone acetyltransferase Tip60 (KAT5) inhibitor with IC50 of 74 uM, with no activity against PCAF and p300. |
