| Cat. No. |
Product Name |
Information |
| PC-61685 |
PU-141
p300/CBP inhibitor
|
PU-141 is a potent, selective CBP/p300 inhibitor that inhibits SK-N-SH cell growth with GI50 of 0.48 uM. |
| PC-60499 |
TH1834 dihydrochloride
Tip60 inhibitor
|
TH1834 dihydrochloride (TH-1834, TH 1834) is a novel potent specific histone acetyltransferase Tip60 inhibitor. |
| PC-60498 |
TH1834
Tip60 inhibitor
|
TH1834 (TH-1834, TH 1834) is a novel potent specific histone acetyltransferase Tip60 inhibitor. |
| PC-70121 |
Windorphen
p300 inhibitor
|
Windorphen is a potent, selective inhibitor of p300 histone acetyltransferase (IC50=4.2 uM). |
| PC-60028 |
A-485
p300/CBP inhibitor
|
A-485 (A485) is a potent, selective and, cell and in vivo active p300/CBP catalytic inhibitor with IC50 of 9.8/2.6 nM. |
| PC-45646 |
I-CBP112
CBP/p300 inhibitor
|
I-CBP112 is a specific and potent inhibitor of CBP/p300 bromodomain with Kd of 150-170 nM. |
| PC-45052 |
Remodelin hydrobromide
NAT10 inhibitor
|
Remodelin hydrobromide is a potent inhibitor of the acetyl-transferase protein NAT10 that acetylates both histones and microtubules. |
| PC-45051 |
Remodelin
NAT10 inhibitor
|
Remodelin is a potent inhibitor of the acetyl-transferase protein NAT10 that acetylates both histones and microtubules. |
| PC-27595 |
CBP/p300 ligand 2
CBP/p300 ligand
|
CBP/p300 ligand 2 is a high affinity ligand of CBP/p300 for PROTAC design. |
| PC-27555 |
CTX-0124143
KAT6A inhibitor
|
CTX-0124143 is a small molecule inhibitor of Monocytic leukemia zinc finger protein (MOZ/KAT6A) with IC50 of 1.0 uM. |
| PC-27554 |
MOZ-IN-3
KAT6A inhibitor
|
MOZ-IN-3 (KAT6A inhibitor 6j) is a potent, selective inhibitor of KAT6A (MOZ, Monocytic leukemia zinc finger protein) with IC50 of 0.03 uM, shows 25-333 fold selectivity against KAT7, KAT5, KAT8 and KAT6B, exhibitsstrong antitumor activity on leukemia cell line K562 (IC50=82 nM). |
| PC-25583 |
Anacardic acid
HAT inhibitor
|
Anacardic acid is a small molecule inhibitor of histone acetyltransferase (HAT) with IC50 of 8.5 and 5.0 uM for p300 and PCAF respectively. |
