| Cat. No. |
Product Name |
Information |
| PC-60639 |
PAT-048
Autotaxin inhibitor
|
PAT-048 (PAT048) is a potent, selective, noncompetitive autotaxin inhibitor with IC50 of 1.1 nM against the lysoPLD activity of human ATX. |
| PC-60638 |
PAT-505
Autotaxin inhibitor
|
PAT-505 (PAT 505, PAT505) is a potent, selective, noncompetitive, and orally active autotaxin inhibitor with IC50 of 2.0 nM against the lysoPLD activity of human ATX. |
| PC-60402 |
GLPG1690
Autotaxin inhibitor
|
GLPG1690 (Ziritaxestat, GLPG 1690) is a first-in-class, potent, competitive autotaxin inhibitor with Ki/IC50 of 15 nM/131 nM. |
| PC-60142 |
BI-2545
Autotaxin inhibitor
|
BI-2545 is a novel potent, selective, orally available Autotaxin inhibitor with IC50 of 2.1 and 3.4 nM for huamn and rat ATX, respectively. |
| PC-45610 |
HA130
Autotaxin inhibitor
|
HA130 (HA-130) is a potent and selective inhibitor of autotaxin with IC50 of 28 nM. |
| PC-23710 |
PAT-505 sodium
Autotaxin inhibitor
|
PAT-505 sodium (PAT 505, PAT505) is a potent, selective, noncompetitive, and orally active autotaxin inhibitor with IC50 of 2.0 nM against the lysoPLD activity of human ATX. |
| PC-23709 |
S32826
Autotaxin inhibitor
|
S32826 is a potent autotaxin inhibitor with IC50 of 8.8 nM, shows similar inhibitory effects at various autotaxin isoforms (α, β and γ), inhibits LPA release from adipocytes. |
| PC-23708 |
BMP22
Autotaxin inhibitor
|
BMP22 is a potent inhibitor of autotaxin (ATX, NPP2) with Ki/IC50 of 0.17/0.27 uM. |
| PC-23707 |
GK442
Autotaxin inhibitor
|
GK442 is a highly potent autotaxin inhibitor with IC50 of 60 nM. |
| PC-23311 |
KR-40795
Autotaxin inhibitor
|
KR-40795 is a novel small molecule autotaxin (ATX) inhibitor with IC50 of 0.13 uM, binds to the allosteric tunnel and hydrophobic pocket of ATX. |
