Vasopressin Receptor (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofVasopressin Receptor Vasopressin Receptor

Cat. No.	Product Name	Information
PC-45460	Conivaptan hydrochloride Vasopressin Receptor inhibitor	Conivaptan (YM-087) is a potent, selective nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively.
PC-45125	Tolvaptan V2R antagonist	Tolvaptan (OPC-41061) is a highly potent selective, competitive vasopressin V2-receptor antagonist with Ki of 0.43 nM, >200-fold more selective than for V1A-receptors.
PC-23097	Invopressin V1a receptor agonist	Invopressin (OCE-205) is a highly selective Vasopressin V1a receptor (V1a receptor) partial agonist (EC50=1.0 nM) with potential for portal hypertension (PHT).
PC-21617	PF-184563 V1a receptor antagonist	PF-184563 is a potent and selective vasopressin V1a antagonist with IC50 of 6.7 nM (hV1a).
PC-21616	Relcovaptan V1a receptor antagonist	SR 49059 (SR-49059) is a potent, selective and orally active vasopressin V1a antagonist with Ki of 1.4 nM.
PC-21615	SRX-246 V1a receptor antagonist	SRX-246 (SRX246) is a potent, selective and CNS penetrant human V1a receptor antagonist with Ki of 0.3 nM.
PC-21614	RGH-122 V1a receptor antagonist	RGH-122 is a potent, selective, and orally bioavailable V1a receptor antagonist with Ki/IC50 of 0.3/0.9 nM (hV1a) respectively, >100-fold selectiive over V2 receptor.
PC-21436	SR-49059 V1AR antagonist	SR49059 (SR-49059) is a potent, selective and orally active vasopressin V1a antagonist with Ki of 1.4 nM.

PREV 12NEXT