| Cat. No. |
Product Name |
Information |
| PC-49652 |
OPC-61815
V2R inhibitor
|
OPC-61815 (Tolvaptan phosphate ester sodium) is a water-soluble phosphate ester pro-drug of Tolvaptan (Cat# PC-45125), which is an orally active vasopressin V2 receptor antagonist. |
| PC-38647 |
Enuvaptan
V1AR antagonist
|
Enuvaptan (BAY2327949) is a potent, selective vasopressin 1a receptor (V1AR) antagonist with potential for renal and cardiovascular diseases. |
| PC-36095 |
Pecavaptan
V1a/V2 receptor antagonist
|
Pecavaptan (BAY 1753011) is a potent, orally active and dual antagonist of vasopressin receptor V1a/V2 receptor (Ki=0.5 nM and 0.6 nM for human, respectively). |
| PC-62116 |
ML389
V1AR antagonist
|
ML389 is a highly potent, selective vasopressin receptor 1a (V1a-R) antagonist with IC50 of 40 nM. |
| PC-61507 |
TASP0434299
V1BR radioligand
|
TASP0434299 is a radioligand candidate for arginine vasopressin 1B (V1B) receptor that exhibits high binding affinities for human and rat V1B receptors with IC50 of 0.526 and 0.641 nM, respectively. |
| PC-70166 |
Conivaptan
Vasopressin Receptor inhibitor
|
Conivaptan (YM-087) is a potent, selective, nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively. |
| PC-60078 |
RG7713
V1a receptor antagonist
|
RG7713 (RO5028442, RG-7713) is a potent, highly selective, brain-penetrant vasopressin 1a (hV1a) antagonist with Ki of 1 nM. |
| PC-60033 |
Balovaptan
V1a receptor antagonist
|
Balovaptan (RG7314, RO5285119) is a potent, selective vasopressin-1 receptor antagonist with Kb of 0.39 nM at the human V1a receptor. |
| PC-47487 |
Ornipressin
|
Ornipressin is a vasoconstrictor, haemostatic and renal agent. |
| PC-45192 |
Desmopressin
V2 receptor antagonist
|
Desmopressin is a synthetic analogue of the antidiuretic hormone arginine vasopressin, binds to V2 receptors in renal collecting ducts, increasing water reabsorption. |
| PC-45191 |
Desmopressin acetate
|
Desmopressin acetate is a synthetic analogue of the antidiuretic hormone arginine vasopressin. |
| PC-45459 |
Mozavaptan
V2 receptor antagonist
|
Mozavaptan (OPC-31260) is a potent, selective nonpeptide vasopressin V2 receptor antagonist with IC50 of 14 nM. |
