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首页-小分子抑制剂&激动剂-GPCR-Vasopressin Receptor-RG7713
RG7713

Chemical Structure : RG7713

CAS No.: 920022-47-5

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RG7713 (RO-5028442;RG-7713;RO5028442)

货号: PC-60078Not For Human Use, Lab Use Only.

RG7713 (RO5028442, RG-7713) is a potent, highly selective, brain-penetrant vasopressin 1a (hV1a) antagonist with Ki of 1 nM.

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5 mg ￥2580 In stock
10 mg ￥3880 In stock
25 mg ￥5580 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

RG7713 (RO5028442, RG-7713) is a potent, highly selective, brain-penetrant vasopressin 1a (hV1a receptor) antagonist with Ki of 1 nM, shows no activiity on hV2 receptor (Ki>30 uM)。
RG7713 (RO5028442) displays moderate mouse affinity and excellent selectivity versus hV2 and hOT receptors.

物理化学性质&存储条件

分子量 437.97
分子式 C25H28ClN3O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(6-Chloro-1-(2-(dimethylamino)ethyl)indol-3-yl)-spiro(1H-isobenzofuran-3,4'-piperidine)-1'-yl-methanone

参考文献

1. Ratni H, et al. J Med Chem. 2015 Mar 12;58(5):2275-89.

2. Umbricht D, et al. Neuropsychopharmacology. 2017 Aug;42(9):1914-1923.

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