Conivaptan hydrochloride |CAS:168626-94-6 Probechem Biochemicals

Chemical Structure : Conivaptan hydrochloride

CAS No.: 168626-94-6

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Conivaptan hydrochloride (YM-087, YM087)

货号: PC-45460Not For Human Use, Lab Use Only.

Conivaptan (YM-087) is a potent, selective nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively.

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50 mg	￥1920	In stock
100 mg	￥3200	In stock
250 mg	￥5900	In stock
1 g		Get quote

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生物&药学活性

Conivaptan (YM-087) is a potent, selective nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively.
Conivaptan (YM-087) is less potent for OT receptors and no effect on V1B receptor.
Conivaptan (YM-087) blocks AVP-induced cAMP production of cultured renal epithelium cells concentration dependently and has no agonistic activities.

物理化学性质&存储条件

分子量	535.0354
分子式	C32H27ClN4O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	[1,1'-Biphenyl]-2-carboxamide, N-[4-[(4,5-dihydro-2-methylimidazo[4,5-d][1]benzazepin-6(1H)-yl)carbonyl]phenyl]-, hydrochloride (1:1)

参考文献

1. Tahara A, et al. J Pharmacol Exp Ther. 1997 Jul;282(1):301-8.

2. Tahara A, et al. Cardiovasc Res. 1998 Apr;38(1):198-205.

3. Nakayama S, et al. Neurocrit Care. 2016 Apr;24(2):273-82.

Conivaptan hydrochloride (YM-087, YM087)

生物&药学活性

物理化学性质&存储条件

参考文献

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Conivaptan hydrochloride (YM-087, YM087)

生物&药学活性

物理化学性质&存储条件

参考文献

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