Mozavaptan (OPC-31260) | V2 receptor antagonist | Probechem Biochemicals

Chemical Structure : Mozavaptan

CAS No.: 137975-06-5

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Mozavaptan (OPC-31260, OPC31260)

货号: PC-45459Not For Human Use, Lab Use Only.

Mozavaptan (OPC-31260) is a potent, selective nonpeptide vasopressin V2 receptor antagonist with IC50 of 14 nM.

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50 mg	￥980	In stock
100 mg	￥1580	In stock
250 mg	￥2580	In stock
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生物&药学活性

Mozavaptan (OPC-31260) is a potent, selective nonpeptide vasopressin V2 receptor antagonist with IC50 of 14 nM.
Mozavaptan 100-fold less potent for VP1 (IC50=1.2 uM).
Mozavaptan dose-dependently increases urine flow and decreases urine osmolality in normal conscious rats; orally effective.

物理化学性质&存储条件

分子量	427.5381
分子式	C27H29N3O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: 6.2 mg/mL (Need warming)
Chemical Name/SMILES	Benzamide, N-[4-[[5-(dimethylamino)-2,3,4,5-tetrahydro-1H-1-benzazepin-1-yl]carbonyl]phenyl]-2-methyl-

参考文献

1. Yamamura Y, et al. Br J Pharmacol. 1992 Apr;105(4):787-91.

2. Tsuboi Y, et al. J Endocrinol. 1994 Nov;143(2):227-34.

3. Wang X, et al. J Am Soc Nephrol. 2005 Apr;16(4):846-51.

Mozavaptan (OPC-31260, OPC31260)

生物&药学活性

物理化学性质&存储条件

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Mozavaptan (OPC-31260, OPC31260)

生物&药学活性

物理化学性质&存储条件

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