SRX-246 | V1a receptor antagonist | Probechem Biochemicals

Chemical Structure : SRX-246

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货号: PC-21615Not For Human Use, Lab Use Only.

SRX-246 (SRX246) is a potent, selective and CNS penetrant human V1a receptor antagonist with Ki of 0.3 nM.

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SRX-246 (SRX246) is a potent, selective and CNS penetrant human V1a receptor antagonist with Ki of 0.3 nM.

分子量	703.88
分子式	C42H49N5O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-4-([1,4'-bipiperidin]-1'-yl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-N-((R)-1-phenylethyl)butanamide

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3. Guillon C, et al. Bioorg Med Chem. 2007;15:2054.