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首页-小分子抑制剂&激动剂-Tyrosine Kinase-Src

Request The Product List ofSrc Src

Cat. No. Product Name Information
PC-45439

KX1-004

Src inhibitor

KX1-004 is a non-ATP competitive Src-PTK inhibitor with IC50 of 40 uM.
PC-42539

KX2-391 mesylate

Src/pretubulin inhibitor

Tirbanibulin mesylate (KX2-391 mesylate) is a highly selective, non-ATP competitive substrate-pocket-directed Src/pretubulin inhibitor.
PC-42538

KX2-391 dihydrochloride

Src inhibitor

Tirbanibulin (KX2-391 dihydrochloride) is a highly selective, non-ATP competitive substrate-pocket-directed Src/pretubulin inhibitor.
PC-42537

KX2-391

Src inhibitor

KX2-391(Tirbanibulin, KX 01, KX 2-391) is a highly selective, non-ATP competitive substrate-pocket-directed Src/pretubulin inhibitor.
PC-25816

DCDBS84 hydrobromide

Integrin β3-Src SH3 inhibitor

DCDBS84 hydrobromide is a small molecule specifically targeting c‐Src SH3 RT‐loop with SPR Kd of 0.83 uM, disrupts the interaction of integrin β3 with Src SH3, selectively blocks αIIbβ3 outside‐in signaling and shows potent antithrombotic effect.
PC-25815

DCDBS84

Integrin β3-Src SH3 inhibitor

DCDBS84 is a small molecule specifically targeting c‐Src SH3 RT‐loop with SPR Kd of 0.83 uM, disrupts the interaction of integrin β3 with Src SH3, selectively blocks αIIbβ3 outside‐in signaling and shows potent antithrombotic effect.
PC-25344

Reynoutrin

Fyn inhibitor

Reynoutrin (Quercetin-3-D-xyloside) is a flavonoid from Psidium cattleianum, with antioxidant and radical-scavenging activity, a potent inhibitor of Fyn, inhibits both the expression and phosphorylation of Fyn.
PC-24574

Src inhibitor PP1

Src inhibitor

PP1 is a potent, selective Src family tyrosine kinases inhibitor with IC50 of 5 and 6 nM for Lck and Fyn, respectively.
PC-24573

Src inhibitor PP2

Src inhibitor

PP2 is a potent, reversible and ATP-competitive Src family kinases inhibitor with IC50 of 4 and 5 nM for Lck and Fyn, respectively, also inhibits RIPK3 with IC50 of 29 nM.
PC-24043

Bosutinib hydrate

Src/Abl inhibitor

Bosutinib hydrate (SKI-606) is a potent, dual Src/Abl inhibitor with IC50 of 1.2 nM (Src enzyme), inhibits Src autophosphorylation with an IC50 of 0.25 uM in HT29 cells, inhibits bacterially expressed Abl kinase activity with IC50 of 1 nM.
PC-24042

Bosutinib

Src/Abl inhibitor

Bosutinib (SKI-606) is a potent, dual Src/Abl inhibitor with IC50 of 1.2 nM (Src enzyme), inhibits Src autophosphorylation with an IC50 of 0.25 uM in HT29 cells, inhibits bacterially expressed Abl kinase activity with IC50 of 1 nM.
PC-22492

(R)-LW-Srci-8

c-Src inhibitor

(R)-LW-Srci-8 is a potent, selective, covalent inhibitor of autophosphorylation site in c-Src kinase with IC50 of 35.83 nM.

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