GPR84 (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-21648	OX04529 GPR84 agonist	OX04529 is a highly potent, selective, G-protein pathway biased and orally bioavailable GPR84 agonist with EC50 of 18.5 pM for inhibition of FSK (25 uM)-induced cAMP production in CHO-hGPR84 cells.
PC-21647	OX04528 GPR84 agonist	OX04528 is a highly potent, selective, G-protein pathway biased and orally bioavailable GPR84 agonist with EC50 of 5.98 pM for inhibition of FSK (25 uM)-induced cAMP production in CHO-hGPR84 cells.
PC-49311	GPR84 inhibitor 42 GPR84 inhibitor	GPR84 inhibitor 42 is a potent GPR84 antagonist with pIC50 of 8.28 in [35S]GTPγS binding assays.
PC-72367	DL-175 GPR84 agonist	DL-175 is a potent and selective biased GPR84 agonist with EC50 of 33 nM.
PC-72361	PSB-17365 GPR84 agonist	PSB-17365 is a potent, selective, Gi-biased agonist of GPR84 with EC50 of 2.5 nM, β-arrestin IC50 of 104 nM in human GPR84-expressing cells.
PC-72360	PSB-1584 GPR84 agonist	PSB-1584 is a potent, selective agonist of GPR84 with EC50 of 5.0 nM, β-arrestin IC50 of 3.2 nM in human GPR84-expressing cells.
PC-72359	PSB-16671 GPR84 agonist	PSB-16671 is a novel orthosteric and allosteric activator of GPR84, activates human GPR84 with EC50 of 41.3 nM in cAMP accumulation assays.
PC-72358	PBI-4547 GPR84 antagonist	PBI-4547 is an agonist of GPR40/120 and an antagonist of GPR84, also is a partial ligand and activator of PPAR.
PC-72357	GPR84 antagonist 837 GPR84 antagonist	Compound 837 (GPR84 antagonist) is a highly potent (affinity, 1 nM), selective antagonist of both orthosteric and allosteric activators of GPR84.
PC-72356	GLPG1205 GPR84 antagonist	GLPG1205 is a potent and selective GPR84 inhibitor (negative allosteric modulator) with IC50 of 54 nM (hGPR84).
PC-43189	6-OAU GPR84 agonist	6-OAU (GTPL5846, 6-n-Octylaminouracil) is a potent, specific agonist of GPR84 with EC50 of 512 nM in [35S]GTPγS binding assay, without activity for GPR109A and OXER1 in a panel of 69 GPCRs.
PC-21649	PSB-16434 GPR84 agonist	PSB-16434 is a highly potent, Gi pathway-selective GPR84 agonist with cAMP EC50 of 7.1 nM, 79-fold selective over β-arrestin-2 recruitment activity.

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