Bombesin Receptor (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-38792	MK-5046 BRS-3 agonist	MK-5046 a potent, selective small molecule agonist of BRS-3 (bombesin receptor subtype-3) with Ki and EC50 values of 3.7 and 14 nM (hBRS-3), respectively.
PC-61219	RC-3095 GRPR (BRS-1) inhibitor	RC-3095 is a potent, peptide bombesin/gastrin releasing peptide (GRPR,BRS-1) antagonist.
PC-61215	Bantag-1 trifluoroacetate	Bantag-1 trifluoroacetate is a potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3.
PC-21220	PD168368 NMB-R antagonist	PD168368 is a potent, competitive, and selective neuromedin B receptor (NMB-R) antagonist with Ki of 15 nM, IC50 of 96 nM.
PC-20957	DSO-5a BRS-3 agonist	DSO-5a (Dimethyl shikonin oxime 5a) is a potent, selective agonist pf bombesin receptor subtype-3 (BB3, BRS-3) with pEC50 of 8.4 (IP-1 accumulation in hBB3-H1299 cells).
PC-61218	BRS-3 agonist Compound A racemate	A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 270/130 nM for human/rat BRS-3, respectively.
PC-61217	(S)-BRS-3 agonist Compound A	The distomer of BRS-3 agonist Compound A, shows no activity for bombesin receptor subtype-3 (BRS-3) with EC50>10 uM..
PC-61216	BRS-3 agonist Compound A	A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 250/100 nM for human/rat BRS-3, resp+H1437+M1438.

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