BRS-3 agonist Compound A racemate

Chemical Structure : BRS-3 agonist Compound A racemate

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货号: PC-61218Not For Human Use, Lab Use Only.

A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 270/130 nM for human/rat BRS-3, respectively.

规格	价格	库存	数量
25 mg		Get quote
100 mg		Get quote
500 mg		Get quote
1 g		Get quote

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生物&药学活性

A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 270/130 nM for human/rat BRS-3, respectively; displays no activity against GRPR (BRS-1) and NMBR (BRS-2) (EC50>10 uM).

物理化学性质&存储条件

分子量	428.532
分子式	C27H28N2O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	6-benzyl-N-tert-butyl-9-methoxy-7-oxo-6,7-dihydro-5H-dibenzo[c,e]azepine-5-carboxamide

参考文献

1. Nio Y, et al. Endocrinology. 2017 May 1;158(5):1298-1313.