Bantag-1 trifluoroacetate

Chemical Structure : Bantag-1 trifluoroacetate

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货号: PC-61215Not For Human Use, Lab Use Only.

Bantag-1 trifluoroacetate is a potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3.

规格	价格	库存	数量
25 mg		Get quote
100 mg		Get quote
500 mg		Get quote
1 g		Get quote

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生物&药学活性

Bantag-1 trifluoroacetate is a potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3.
Bantag-1 trifluoroacetate displays 1000-fold selectivity over hNMBR and hGRPR.
Bantag-1 trifluoroacetate increases food intake and produces an obesity phenotype in mice.

物理化学性质&存储条件

分子量
分子式	C48H73N8O7 · xC2HF3O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Boc-Phe-His-4-amino-5-cyclohexyl-2,4,5-trideoxypentonyl-Leu-(3-dimethylamino) benzylamide N-methylammonium trifluoroacetate salt

参考文献

1. Moreno P, et al. J Pharmacol Exp Ther. 2013 Oct;347(1):100-16.

2. Guan XM, et al. Cell Metab. 2010 Feb 3;11(2):101-12.

3. Feng Y, et al. Endocrinology. 2011 Nov;152(11):4106-15.

4. Nakamura T, et al. Biochem Pharmacol. 2016 Sep 1;115:64-76.