| Cat. No. |
Product Name |
Information |
| PC-20101 |
GS-6201
A2BR antagonist
|
GS-6201 (CVT-6883, GS-6201) is a specific and selective A2B adenosine receptor antagonist with Ki of 22 nM, >50-fold selectivity over A3, A1 and A2A receptors. |
| PC-20100 |
JNJ-40255293
Adenosine A2A/A1 inhibitor
|
JNJ-40255293 (JNJ 40255293) is a potent, dual adenosine A2A/A1 receptor antagonist with Ki of 6.8/42 nM, respectively. |
| PC-49545 |
PSB-603
A2BR antagonist
|
PSB-603 is a potent, selective adenosine A2B receptor antagonist with Ki of 0.553 nM, >17000-fold selectivity over other adenosine receptors (A1, A2A and A3 receptors). |
| PC-49354 |
M1069
A2AR/A2BR antagonist
|
M1069 (M-1069) is a potent, dual antagonist of the A2A and A2B adenosine receptors, with selectivity of >100 fold against the A1 and A3 receptors. |
| PC-49105 |
BnOCPA
A1R agonist
|
BnOCPA is a potent and powerful analgesic and a highly selective and potent, full agonist at human adenosine A1 receptors (A1Rs) with pEC50 of 7.23 in a NanoBRET agonist binding assay. |
| PC-38488 |
CGS-15943
Adenosine receptor inhibitor
|
CGS-15943 is a potent, non-xanthine adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively. |
| PC-38365 |
Inupadenant
A2AR antagonist
|
Inupadenant (EOS-850, EOS100850) is a non brain-penetrant, potent and highly selective small molecule antagonist of adenosine A2a receptor (A2AR), shows activity at the high adenosine concentrations found in tumors. |
| PC-38014 |
MIPS521
A1R modulator
|
MIPS521 (MIPS-521) is a potent, positive allosteric modulator (PAM) of adenosine A1 receptor (A1AR). |
| PC-36101 |
KH-176
ROS-redox modulator
|
KH-176 (KH176, Sonlicromanol) is a smal molecule ROS-redox modulator, effectively reduces increased cellular ROS levels and protects OXPHOS deficient primary cells against redox perturbation by targeting the Thioredoxin/Peroxiredoxin system. |
| PC-35973 |
MRS1186
A3AR antagonist
|
MRS1186 (MRS-1186) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist with Ki of 7.66 nM.. |
| PC-35841 |
AB928
Adenosine receptor inhibitor
|
Etrumadenant (AB928) is a potent, dual antagonist of the A2aR and A2bR adenosine receptors with Kb of 1.5 and 2.0 nM, respectively. |
| PC-35779 |
PBF509
A2AR antagonist
|
PBF509 (Taminadenant, PBF-509, NIR 178) is a novel selective and potent Adenosine A2A Receptor (A2AR) antagonist, antagonizes A2AR agonist-mediated cAMP accumulation and impedance responses with KB values of 72.8 and 8.2 nM, respectively. |
