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首页-小分子抑制剂&激动剂-GPCR-Adenosine Receptor-MRS7935
MRS7935

Chemical Structure : MRS7935

CAS No.:

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MRS7935 (MRS 7935)

货号: PC-21510Not For Human Use, Lab Use Only.

MRS7935 is a potent, selective positive allosteric modulator (PAM) of A1 adenosine receptor (A1AR) with EC50 of 1.43 uM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    MRS7935 is a potent, selective positive allosteric modulator (PAM) of A1 adenosine receptor (A1AR) with EC50 of 1.43 uM.
    MRS7935 displays no functional activity at hA2A, hA2B, and hA3ARs at 30 μM.
    MRS7935 (1 uM) enhances the functional activity of A1AR agonist Cl-ENBA.
    MRS7935 does not enhance hypothermia in vivo induced by either adenosine or a selective A1AR agonist.

    物理化学性质&存储条件

    分子量 443.94
    分子式 C24H20ClF2NOS
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (2-amino-5-((3,4-difluorophenyl)ethynyl)-4-neopentylthiophen-3-yl)(4-chlorophenyl)methanone

    参考文献

    1. Paola Oliva, et al. ACS Medicinal Chemistry Letters, 2023.

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