TRR469 | A1AR modulator | Probechem Biochemicals

Chemical Structure : TRR469

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TRR469 (TRR-469, TRR 469)

货号: PC-21513Not For Human Use, Lab Use Only.

TRR469 is a potent, selective adenosine A1 receptor (A1AR) positive allosteric modulator with pKb of 5.36, exhibits anti-nociceptive properties in acute and neuropathic pain models in mice.

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生物&药学活性

TRR469 is a potent, selective adenosine A1 receptor (A1AR) positive allosteric modulator with pKb of 5.36, exhibits anti-nociceptive properties in acute and neuropathic pain models in mice.

物理化学性质&存储条件

分子量	506.04
分子式	C28H25ClFN3OS
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(2-Amino-4-[(4-(phenyl)piperazin-1-yl)methyl]-5-(4-fluorophenyl)thiophen-3-yl)-(4-chlorophenyl)methanone

参考文献

1. Vincenzi F, et al. Neuropharmacology. 2016 Dec;111:283-292.

2. Romeo Romagnoli, et al. J Med Chem. 2012 Sep 13;55(17):7719-35.

TRR469 (TRR-469, TRR 469)

生物&药学活性

物理化学性质&存储条件

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TRR469 (TRR-469, TRR 469)

生物&药学活性

物理化学性质&存储条件

参考文献

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