| Cat. No. |
Product Name |
Information |
| PC-42717 |
Vipadenant
A2AR antagonist
|
Vipadenant (BIIB014) is a potent and selective A2A adenosine receptor antagonist with Ki of 1.3 nM. |
| PC-42729 |
Preladenant
A2AR antagonist
|
Preladenant (SCH420814) is a potent and highly selective adenosine A2A receptor competitive antagonist with Ki of 1.1 nM. |
| PC-42728 |
Istradefylline
A2AR antagonist
|
Istradefylline (KW6002) is a potent and highly selective A2A receptor antagonist with Ki of 2.2 nM. |
| PC-45527 |
APNEA
A3AR agonist
|
APNEA is a non-selective agonist of adenosine A3 receptor, has a high affinity for the adenosine A1 and A3 receptors. |
| PC-45624 |
AB-MECA
A3AR agonist
|
AB-MECA is a high affinity A3 adenosine receptor (A3AR) agonist with binding Ki of 430.5 nM for human A3 receptors in CHO cells. |
| PC-24291 |
HZ-086
A2AR inhibitor
|
HZ-086 is a potent and selective inhibitor of adenosine A2A receptor (A2AR) with Ki of 1.4 nM (hA2A), >250-fold selective over A1R and A3R. |
| PC-24196 |
Zaladenant
A2a receptor inhibitor
|
Zaladenant is a potent, selective adenosine A2a receptor inhibitor with IC50 of 0.23 nM. |
| PC-23909 |
FM101
A3AR inhibitor
|
FM101 is a highly potent and selective antagonist of A3 adenosine receptor (A3AR), selectively binds to human A3AR with Ki of 1.44 nM. |
| PC-23655 |
Regadenoson
A2A receptor antagonist
|
Regadenoson (CVT-3146) is a potent, selective A2A adenosine receptor agonist, and short-acting coronary vasodilator. |
| PC-23389 |
SLV320
Adenosine A1 receptor antagonist
|
Derenofylline (SLV320) is a potent, selective and orally active adenosine A1 receptor antagonist with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. |
| PC-23365 |
TC-G 1004
A2A receptor antagonist
|
TC-G 1004 is a potent, selective orally active A2A adenosine receptor (A2A R) antagonist, with Ki values of 0.44 nM and 80 nM for hA2A and hA1, respectively. |
| PC-22840 |
DPCPX
Adenosine A1 receptor antagonist
|
DPCPX (PD116948) is a highly potent and selective adenosine A1 receptor antagonist with Ki of 0.46 nM, >500-fold selective over A2 receptor. |
