eN-IN-1 |CAS:95523-13-0 Probechem Biochemicals

Chemical Structure : eN-IN-1

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eN-IN-1 (N-[(4-Aminophenyl)methyl]adenosine)

货号: PC-42064Not For Human Use, Lab Use Only.

An α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 29 nM for rat recombinant eN.

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生物&药学活性

eN-IN-1 (N-[(4-Aminophenyl)methyl]adenosine) is an α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 29 nM for rat recombinant eN.
eN-IN-1 also exhibits dual-action properties toward both A2AR and equilibrative nucleoside transporter 1 (ENT1) with Ki of 27.7 uM and 6.51 nM.

物理化学性质&存储条件

分子量	372.3785
分子式	C17H20N6O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Adenosine, N-[(4-aminophenyl)methyl]-

参考文献

1. Bhattarai S, et al. J Med Chem. 2015 Aug 13;58(15):6248-63.

2. Chen JB, et al. ChemMedChem. 2011 Aug 1;6(8):1390-400.

eN-IN-1 (N-[(4-Aminophenyl)methyl]adenosine)

生物&药学活性

物理化学性质&存储条件

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eN-IN-1 (N-[(4-Aminophenyl)methyl]adenosine)

生物&药学活性

物理化学性质&存储条件

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