Glycine Transporter (GlyT) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofGlycine Transporter (GlyT) Glycine Transporter (GlyT)

Cat. No.	Product Name	Information
PC-60526	Opiranserin GlyT2 inhibitor	Opiranserin (VVZ-149, VVZ-000149) is a potent, selective, mixed glycine GlyT2 transporter blocker (IC50= 0.86 uM), purine P2X3 receptor antagonist (IC50=0.87 uM) and serotonin 5-HT2A receptor antagonist (IC50=1.3 uM).
PC-60446	ALX-1393 GlyT2 inhibitor	ALX-1393 (ALX 1393, ALX1393) is a potent, specific GlyT2 inhibitor with Ki of <1 uM.
PC-60445	Org 25543 GlyT2 inhibitor	Org 25543 is a potent, highly selective glycine transporter 1 (GlyT2) inhibitor with IC50 of 16 nM with negligible affinity for GlyT1.
PC-60444	Org 25935 GlyT1 inhibitor	Org 25935 (SCH 900435) is a potent, selective glycine transporter 1 (GlyT1) inhibitor with IC50 of 100 nM.
PC-42145	LY2365109 hydrochloride GlyT1 inhibitor	LY2365109 hydrochloride is a potent and selective GlyT1 inhibitor with IC50 of 15.8 nM, displays no activity for GlyT2 (IC50>30 uM).
PC-42706	Bitopertin GlyT1 inhibitor, Nrf2 activator	Bitopertin (RG1678, RO4917838) is a potent and selective glycine uptake GlyT1 inhibitor with EC50 of 30 nM, also is an Nrf2 activator.
PC-42707	Bitopertin R enantiomer	A potent and selective GlyT1 inhibitor with EC50 of 54 nM.

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