Org 25543 |CAS:495076-64-7 Probechem Biochemicals

Chemical Structure : Org 25543

CAS No.: 495076-64-7

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货号: PC-60445Not For Human Use, Lab Use Only.

Org 25543 is a potent, highly selective glycine transporter 1 (GlyT2) inhibitor with IC50 of 16 nM with negligible affinity for GlyT1.

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Org 25543 is a potent, highly selective glycine transporter 1 (GlyT2) inhibitor with IC50 of 16 nM with negligible affinity for GlyT1.

分子量	448.988
分子式	C24H33ClN2O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Benzamide, N-[[1-(dimethylamino)cyclopentyl]methyl]-3,5-dimethoxy-4-(phenylmethoxy)-, monohydrochloride (9CI)

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2. Rousseau F, et al. J Neurosci. 2008 Sep 24;28(39):9755-68.

3. Romei C, et al. J Neurochem. 2011 Oct;119(1):50-63.

4. Mingorance-Le Meur A, et al. Br J Pharmacol. 2013 Nov;170(5):1053-63.